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Catalog name Description price
R-R-3968 Carvedilol (Standard) CAS No.72956-09-3 Carvedilol (Standard)/CAS No.72956-09-3 is the analytical standard of Carvedilol. This product is intended for research and analytical applications. Carvedilol (BM 14190) is a non-selective β/α-1 blocker. Carvedilol inhibits lipid peroxidation in a dose-dependent manner with an IC50 of 5 μM. Carvedilol is a multiple action antihypertensive agent with potential use in angina and congestive heart failure. Carvedilol is an autophagy inducer that inhibits the NLRP3 inflammasome. price>
R-R-3969 Betaxolol-d5 CAS No.1189957-99-0 Betaxolol-d5/CAS No.1189957-99-0 is the deuterium labeled Betaxolol. Betaxolol is a selective beta1 adrenergic receptor blocker that can be used for the research of hypertension and glaucoma. price>
R-R-3970 HEAT hydrochloride CAS No.30007-39-7 HEAT (BE2254) hydrochloride/CAS No.30007-39-7 is a selective alpha 1 adrenergic receptor antagonist. HEAT hydrochloride, a phenethylamine derivative, shows pKis of 9, 9.1, and 8.57 for alpha 1a, alpha 1b and alpha 1c, respectively. price>
R-R-3971 RS100329 hydrochloride CAS No.1215654-26-4 RS100329 hydrochloride/CAS No.1215654-26-4 is a potent and selective α1A-adrenoceptor antagonist with pKi values of 9.6, 7.9 and 7.5 for α1A, α1D, and α1B, respectively. RS100329 hydrochloride inhibits reflex urethral contractions. RS100329 hydrochloride can be used in research of benign prostatic hyperplasia. price>
R-R-3972 Agroclavine CAS No.548-42-5 Agroclavine/CAS No.548-42-5 is a natural, clavine type of ergot alkaloid. Agroclavine is a D1 dopamine receptor and α1-adrenoceptor agonist. Agroclavine also has anticancer and antimicrobial activities. price>
R-R-3973 Brombuterol hydrochloride CAS No.21912-49-2 Brombuterol hydrochloride (Bromobuterol hydrochloride)/CAS No.21912-49-2 is a β-adrenergic receptor agonist. price>
R-R-3974 (Rac)-Nebivolol CAS No.99200-09-6 (Rac)-Nebivolol ((Rac)-R 065824)/CAS No.99200-09-6 is a racemic isomer of Nebivolol. Nebivolol is a selective β1-adrenergic receptor antagonist with an IC50 value of 0.8 nM. Nebivolol can prevent up-regulation of Nox2/NADPH oxidase and lipoperoxidation in the early stages of ethanol-induced cardiac toxicity. Vasodilatory activity. price>
R-R-3975 Terbutaline sulfate (Standard) CAS No.23031-32-5 Terbutaline (sulfate) (Standard)/CAS No.23031-32-5 is the analytical standard of Terbutaline (sulfate). This product is intended for research and analytical applications. Terbutaline sulfate is an orally active β2-adrenergic receptor agonist and an active metabolite of bambuterol. Terbutaline sulfate can be used in asthma symptom research. price>
R-R-3976 Isoxsuprine-d6 hydrochloride CAS No.2706004-35-3 Isoxsuprine-d6 (hydrochloride)/CAS No.2706004-35-3 is the deuterium labeled Isoxsuprine hydrochloride. Isoxsuprine hydrochloride is a beta-adrenergic receptor agonist with Kis of 13.65 μΜ and 3.48 μΜ for myometrial and placcntal beta-adrenergic receptor, respectively. Isoxsuprine hydrochloride is also a NMDA receptor antagonist. price>
R-R-3977 Azepexole dihydrochloride CAS No.36067-72-8 Azepexole (B-HT 933) dihydrochloride/CAS No.36067-72-8 is a potent and selective alpha 2-adrenoceptor agonist with pKis of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions (IC50= 78.72 nM). price>