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Home > products > apis> gpcr-g-protein
Catalog name Description price
R-R-4021 GSK1820795A CAS No.2650253-86-2 GSK1820795A/CAS No.2650253-86-2, as a telmisartan analog, is a selective hGPR132a antagonist. GSK1820795A blocks activation of yeast cells expressing hGPR132a by N-acylamides. GSK1820795A is also a angiotensin II antagonists and partial PPARγ agonists (compound 38). price>
R-R-4022 Azilsartan-d5 CAS No.1346599-45-8 Azilsartan-d5/CAS No.1346599-45-8 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. price>
R-R-4023 Irbesartan-d4 CAS No.1216883-23-6 Irbesartan-d4/CAS No.1216883-23-6 is the deuterium labeled Irbesartan, which is a highly potent and specific angiotensin II type 1 (AT1) receptor antagonist. price>
R-R-4024 Telmisartan-d3 CAS No.1189889-44-8 Telmisartan-d3/CAS No.1189889-44-8 is the deuterium labeled Telmisartan. Telmisartan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM. price>
R-R-4025 Eprosartan mesylate CAS No.144143-96-4 Eprosartan mesylate (SKF-108566J)/CAS No.144143-96-4 is a selective, competitive, nonpeptid and orally active angiotensin II receptor antagonist, used as an antihypertensive. Eprosartan mesylate binds angiotensin II receptor with IC50s of 9.2 nM and 3.9 nM in rat and human adrenal cortical membranes, respectively. price>
R-R-4026 Candesartan-d4 CAS No.1346604-70-3 Candesartan-d4/CAS No.1346604-70-3 is the deuterium labeled Candesartan, which is an angiotensin II receptor antagonist. price>
R-R-4027 Olmesartan lactone impurity CAS No.849206-43-5 Olmesartan lactone impurity/CAS No.849206-43-5 is a cyclic ester impurity of Olmesartan. Olmesartan is an angiotensin II receptor (AT1R) antagonist and has the potential for high blood pressure study. price>
R-R-4028 Losartan-d4 (carboxylic acid) CAS No.1246820-62-1 Losartan-d4 (carboxylic acid)/CAS No.1246820-62-1 is the deuterium labeled Losartan (EXP-3174), which is an angiotensin II receptor antagonist. price>
R-R-4029 Angiotensin II (5-8), human Angiotensin II (5-8), human is an endogenous C-terminal fragment of the peptide vasoconstrictor angiotensin II. Angiotensin II binds the AT II type 1 (AT1) receptor, stimulating GPCRs in vascular smooth muscle cells and increasing intracellular Ca2+ levels. Angiotensin II also acts at the Na+/H+ exchanger in the proximal tubules of the kidney. price>
R-R-4030 Losartan-d4 CAS No.1030937-27-9 Losartan-d4/CAS No.1030937-27-9 is the deuterium labeled Losartan. Losartan is an angiotensin II receptor antagonist, competing with the binding of angiotensin II to AT1 receptors with IC50 of 20 nM. price>