Product apis-dna-damage-dna-repa

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Catalog	name	Description	price
R-R-4490	CK2/ERK8-IN-1 CAS No.1085822-09-8	CK2/ERK8-IN-1/CAS No.1085822-09-8 is a dual casein kinase 2 (CK2) (Ki of 0.25 µM) and ERK8 (MAPK15, ERK7) inhibitor with IC50s of 0.50 μM. CK2/ERK8-IN-1 also binds to PIM1, HIPK2 (homeodomain-interacting protein kinase 2), and DYRK1A with Kis of 8.65 µM, 15.25 µM, and 11.9 µM, respectively. CK2/ERK8-IN-1 has pro-apoptotic efficacy.	price>
R-R-4491	Epiblastin A CAS No.16470-02-3	Epiblastin A/CAS No.16470-02-3 is an ATP competitive casein kinase 1 (CK1) inhibitor with IC50s of 8.9, 0.5, and 4.7 µM for CK1α, CK1δ, and CK1 ɛ, respectively. Epiblastin A induces reprogramming of epiblast stem cells into embryonic stem cells by inhibition of CK1.	price>
R-R-4492	MRT00033659 CAS No.1401731-54-1	MRT00033659/CAS No.1401731-54-1 is a potent broad-spectrum kinase inhibitor of CK1 (IC50=0.9 µM for CK1δ) and CHK1 (IC50=0.23 µM). MRT00033659, a pyrazolo-pyridine analogue, induces p53 pathway activation and E2F-1 destabilisation.	price>
R-R-4493	TMX-4113 CAS No.2766385-92-4	TMX-4113/CAS No.2766385-92-4 is a degrader of phosphodiesterase 6D (PDE6D) and casein kinase 1α (CK1α). TMX-4113 can be used for the research of cancer.	price>
R-R-4494	LH846 CAS No.639052-78-1	LH846/CAS No.639052-78-1 is a selective inhibitor of CKIδ, with an IC50 of 290 nM, and less potently inhibits CKIα and CKIε, with IC50s of 2.5 μM and 1.3 μM, respectively.	price>
R-R-4495	Casein Kinase II Inhibitor IV CAS No.863598-09-8	Casein Kinase II Inhibitor IV/CAS No.863598-09-8 is a potent, ATP-competitive of casein kinase II inhibitor with an IC50 of 9 nM. Casein Kinase II Inhibitor IV ia also a human keratinocytes (NHEK) differentiation inducer.	price>
R-R-4496	MU1742	MU1742 is a probe for CK1δ and CK1ε protein kinases.	price>
R-R-4497	PI-828 CAS No.942289-87-4	PI-828/CAS No.942289-87-4 is a dual PI3K and casein kinase 2 (CK2) inhibitor with IC50s of 173 nM, 149 nM, and 1127 nM for p110α, CK2, and CK2α2 in lipid kinase assay, respectively.	price>
R-R-4498	Casein Kinase 2 Substrate Peptide CAS No.132176-35-3	Casein Kinase 2 Substrate Peptide is a common CK2 substrate peptide. Casein Kinase 2 Substrate Peptide is synthesized with its C-terminus conjugated to 5-[(2-aminoethyl)amino]naphthalene-1-sulfonic acid (EDANS). Casein Kinase 2 Substrate Peptide can be used for protein kinase CK2 activity determination.	price>
R-R-4499	CK2 inhibitor 2 CAS No.2641079-92-5	CK2 inhibitor 2/CAS No.2641079-92-5 is a potent, selective and orally active inhibitor of CK2, with an IC50 of 0.66 nM. CK2 inhibitor 2 shows high selectivity for Clk2 (IC50=32.69 nM)/CK2. CK2 inhibitor 2 exhibits favorable antiproliferative and antitumor activity.	price>

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