Product apis-ubiquitin

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Catalog	name	Description	price
R-C-3115	DUBs-IN-2 CAS：924296-19-5	DUBs-IN-2 is a potent deubiquitinase enzyme inhibitor with IC50s of 7.2uM/0.93uM for USP7/USP8 respectively.	price>
R-C-3116	HBX 41108 CAS：924296-39-9	HBX 41108 is an inhibitor of ubiquitin-specific protease (USP)7 activity(IC50=424nM).	price>
R-C-3117	GNE-490 CAS：1033739-92-2	GNE-490 is a highly selective pan-PI3K inhibitor that demonstrates selectivity over mTOR.	price>
R-C-3119	Vialinin A CAS：858134-23-3	Vialinin A is a terphenyl compound originally isolated from the fungi T. terrestris and T.vialis.	price>
R-C-3120	MSC1094308 CAS:2219320-08-6	MSC1094308 is a reversible and allosteric inhibitor of the type II AAA ATPase human ubiquitin-directed unfoldase(VCP)/p97 and the type I AAA ATPase VPS4B,with IC50 values of 0.71μM and 7.2μM for VPS4B and p97,respectively.	price>
R-C-3121	NMS-859 CAS:1449236-96-7	NMS-859 is a potent,covalent VCP(p97)inhibitor,with IC50s of 0.37 and 0.36μM for wild-type VCP in the presence of 60μM and 1 mM ATP in cells,respectively.	price>
R-C-3122	ML241 CAS:1346528-06-0	ML241 is a potent and selective inhibitors of p97 ATPase. ML241 inhibit p97 ATPase with IC(50) values of 100 nM. ML241 inhibits degradation of a p97-dependent but not a p97-independent proteasome substrate in a dual-reporter cell line.	price>
R-C-3123	SR-2211 CAS:1359164-11-6	SR-2211 selectively binds RORr(Ki=105nM),acting as an inverse agonist of constitutive in vitro RORr activity (IC50=320nM).	price>
R-C-3124	AGN-242428(Vimirogant,VTP-43742) CAS:1802706-04-2	AGN-242428,also known as VTP-43742,is a potent,selective and orally active RORγt inhibitor for the treatment of autoimmune disorders,including multiple sclerosis and psoriasis.	price>
R-C-3129	A-9758 CAS:2055271-22-0	A-9758 is a RORγ ligand and a potent,selective RORγt inverse agonist (IC50=5nM),and exhibits robust potency against IL-17A release.	price>

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