Product apis-neuronal-signaling

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Catalog	name	Description	price
R-C-2395	Silodosin CAS:160970-54-7	Silodosin(KAD 3213;KMD 3213)is a potent,selective and orally active α1A-adrenergic receptor(α1A-AR)blocker.Silodosin is an effective and well-tolerated agent,it can be used for the investigation of LUTS/BPH.	price>
R-C-2396	Nebivolol hydrochloride (R-65824) CAS:152520-56-4	Nebivolol hydrochloride selectively inhibits β1- adrenergic receptor with IC50 of 0.8nM.	price>
R-C-2397	BMY 7378 Dihydrochloride CAS:21102-95-4	BMY 7378 is a multi-targeted inhibitor of α2C-adrenoceptor and α1D-adrenoceptor with pKi of 6.54 and 8.2,respectively,and acts as a mixed agonist and antagonist for 5-HT1A receptor with pKi of 8.3.	price>
R-C-2399	Naftopidil CAS:57149-07-2	Naftopidil(KT-611)is is a selective alpha1-adrenoceptor antagonist,with Kis of 3.7nM,20nM and 1.2nM for the cloned human α1a-,α1b-and α1d-adrenoceptor subtypes,respectively.Naftopidil has antiproliferative effects.Naftopidil can be used for the research of prostate hyperplasia.	price>
R-C-2400	Timolol Maleate CAS:26921-17-5	(S)-Timolol Maleate(L-714,465 Maleate)is a non-cardioselective hydrophilic β-adrenoceptor blocker.(S)-Timolol Maleate is widely used as standard medication for intraocular pressure(glaucoma)by preventing the production of aqueous humor. (S)-Timolol Maleate can be used for hypertension,angina pectoris and myocardial infarction.	price>
R-C-2401	Fargesin CAS:31008-19-2	Fargesin is a lignan from Magnolia fargesii,an oriental medicine used in the treatment of nasal congestion and sinusitis.Fargesin exhibits anti-inflammation effects on THP-1 cells via suppression of PKC pathway including downstream JNK, nuclear factors AP-1 and NF-ĸB.	price>
R-C-2402	Dapiprazole Hydrochloride CAS:72822-13-0	Dapiprazole Hydrochloride(Glamidolo Hydrochloride,Reversil Hydrochloride)is the hydrochloride salt form of dapiprazole,an alpha-adrenergic blocker used to reverse mydriasis after eye examination.	price>
R-C-2404	Piribedil CAS:3605-01-4	Piribedil(Trivastal,Trivastan)is a relatively selective dopamine(D2/D3)agonist with moderate antidepressant activity.It also has α2-adrenergic(α2A/α2C)antagonist properties.	price>
R-C-2407	Desvenlafaxine CAS:93413-62-8	Desvenlafaxine is a synthetic form of the major active metabolite of venlafaxine (sold under the brand names Effexor and Efexor).It is being targeted as the first non-hormonal based treatment for menopause.Desvenlafaxine is a synthetic phenethylamine bicyclic derivative with antidepressant activity. Desvenlafaxine is a selective reuptake inhibitor of serotonin and norepinephrine due to its high binding affinities to the pre-synaptic serotonin and norepinephrine transporters.	price>
R-C-2408	Esmolol CAS:81147-92-4	Esmolol is a short acting hyperselective β-adrenergic blocker effective in blunting adrenergic response to several perioperative stimuli and so it might interfere in the effect of the anesthetic drugs on the brain.Esmolol is effective not only in attenuating intraoperative hemodynamic changes related to sympathetic overdrive but also in minimizing significant propofol and sevoflurane requirements without compromising the hemodynamic status.	price>

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