Product apis-Inhibitor-customization

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Catalog	name	Description	price
R-C-2244	Pectolinarin CAS： 28978-02-1	Pectolinarin is a Cirsium isolate with anti-inflammatory activity and similar in chemical structure to linarin.	price>
R-C-2494	PTZ-343 CAS:101199-38-6	PTZ-343 is a potent enhancer of Luminol(HY-15922).PTZ-343 greatly increases the light output of the peroxidase-catalyzed luminol chemiluminescent oxidation reaction(>80%).	price>
R-C-2495	Golotimod CAS ：229305-39-9	Golotimod (SCV-07),an immunomodulating peptide with antimicrobial activity, significantly increases the efficacy of antituberculosis therapy,stimulates thymic and splenic cell proliferation,and improves macrophage function.Golotimod(SCV-07)inhibits STAT3 signaling and modulates the duration and severity of oral mucositis in animal models that received radiation or a combination of radiation and Cisplatin.	price>
R-C-2698	Tautomycetin CAS：119757-73-2	Tautomycetin is a potent and specifical PP1 inhibitor with the potential apoptosis-inducing activity.Tautomycetin inhibits purified PP1 and PP2A enzymes with IC50s of 1.6nM and 62nM,respectively.Tautomycetin is an antifungal antibiotic and has immunosuppressive effects in vivo.	price>
R-C-2728	Zardaverine CAS：101975-10-4	Zardaverine is a newly developed dual-selective PDE3/4 inhibitor with IC50 values of 0.5 uM and 0.8uM respectively.	price>
R-C-2966	Etoricoxib CAS：202409-33-4	Etoricoxib is a synthetic, nonsteroidal anti-inflammatory drug (NSAID) with antipyretic, analgesic, and potential antineoplastic properties. Etoricoxib specifically binds to and inhibits the enzyme cyclooxygenase-2 (COX-2), resulting in inhibition of the conversion of arachidonic acid into prostaglandins. Inhibition of COX-2 may induce apoptosis and inhibit tumor cell proliferation and angiogenesis.	price>
R-C-2971	Lumiracoxib CAS:220991-20-8	Lumiracoxib is a novel, selective COX-2 inhibitor with IC50 and Ki of 0.14 μM and 0.06 μM, exhibits 515-fold selectivity over COX-1. Only for scientific research, not for human body.	price>
R-C-2974	NPS 2390 CAS:226878-01-9	NPS2390 is a group I mGlu antagonist. It displays noncompetitive antagonist activity at both mGlu1 and mGlu5 receptors. NPS2390 is thought to act on a site separate from the glutamate binding pocket.Only for scientific research, not for human body.	price>
R-C-2975	Lofepramine CAS# 23047-25-8	Lofepramine is a first generation tricyclic antidepressant. Lofepramine is a serotonin and noradrenaline re-uptake inhibitor (SNRI) that is metabolized to desipramine (sc-200158, sc-207535).Only for scientific research, not for human body.	price>
R-C-2984	Ro 28-1675 CAS:300353-13-3	Ro 28-1675 (Ro 0281675) is a potent allosteric GK activator with a SC1.5 value of 0.24,0.0019 uM.Only for scientific research, not for human body.	price>

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