Product apis-Inhibitor-customization

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Catalog	name	Description	price
R-R-0330	DCL (PSMA inhibitor) (ACUPA)	DCL (PSMA inhibitor) (ACUPA) is an amino-modified amino acid and a new type of inhibitor that has a highly inhibitory effect on prostate-specific membrane antigen (PSMA). It is introduced into polypeptides through chemical synthesis, thereby changing the properties and activity of the polypeptide. ACUPA-modified amino groups have stability and water solubility, which can enhance the affinity and selectivity of peptides, thereby improving the efficacy and biological activity of peptides. It can also alter the metabolism and distribution of peptides.	price>
R-R-1077	12-O-Methylcarnosic acid	12-O-Methylcarnosic acid (12-Methoxycarnosic acid)/Cas No.62201-71-2, a diterpene carnosic acid isolated from the acetone extract of Salvia microphylla, is an active constituent of 5α-reductase inhibition with an IC50 value of 61.7 μM.	price>
R-M-435	IMT1B	IMT1B (LDC203974) is an orally active, noncompetitive and specific allosteric inhibitor of mitochondrial RNA polymerase (POLRMT) and inhibits mitochondrial DNA (mtDNA) expression. IMT1B has anti-tumour effects.	price>
R-C-590	Dabigatran etexilate cas:872728-81-9	Dabigatran etexilate(BIBR 1048)is an orally active prodrug of Dabigatran. Dabigatran etexilate has anticoagulant effects and is used for the prophylaxis of venousthromboembolism and stroke due to atrial fibrillation.	price>
R-C-612	PluriSln 1 cas:91396-88-2	stearoyl-CoA desaturase 1(SCD1)inhibitor.Used to selectively eliminate undifferentiated human pluripotent stem cells(hPSCs)from culture;induces ER stress,attenuates protein synthesis and induces apoptosis in hPSCs.Prevents teratoma formation in immunocompromised mice.	price>
R-C-623	GSK2838232A cas:1443461-21-9	GSK2838232, a betulin derivative,is an inhibitor of human immune virus (HIV) maturation which is potential for the treatment of chronic HIV infection.	price>
R-C-633	sp-420 cas:1221411-72-8	SP-420 is an orally active small molecule that selectively binds iron and removes it from the body.In animal studies,SP-420 has shown excellent tissue penetration, highly efficient iron binding and a promising safety profile.	price>
R-C-640	Pirodavir cas:124436-59-5	Pirodavir is a potent,broad-spectrum picornavirus inhibitor,and is highly active against both group A and group B rhinovirus serotypes.Pirodavir is very potent in a virus yield reduction assay(IC90=2.3 nM).	price>
R-C-857	5-hydroxydopamine-cisplatin-5-hydroxydopamine	Cisplatin(CDDP)is a platinum containing anticancer drug,namely CIS dichlorodiamine combined with platinum(II).Its brownish yellow powder is a cell cycle nonspecific drug.It has therapeutic effect on sarcoma,malignant epithelial tumor,lymphoma and germ cell tumor.	price>
R-C-877	BMS-1（HY19991） CAS:1675201-83-8	BMS-1(PD-1/PD-L1 inhibitor1,PD1-PDL1-IN1)is a small-molecule inhibitor of PD-1/PD-L1 interaction with IC50 of 6 nM.	price>

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