Product apis-membranet-transporters

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Catalog	name	Description	price
R-C-3249	TRPC6-IN-1 CAS:901715-05-7	TRPC6-IN-1 is a Transient Receptor Potential Canonical 6 Channel (TRPC6) inhibitor, with an EC50 of 4.66 μM.Our products are only suitable for scientific research experiments, not for clinical experiments and human body.	price>
R-C-3250	Pico145 CAS:1628287-16-0	Pico145 is a remarkable inhibitor of TRPC1/4/5 channels,inhibits-englerin A-activated TRPC4/TRPC5 channels,with IC50s of 0.349 and 1.3nM in cells,and shows no effect on TRPC3,TRPC6,TRPV1,TRPV4,TRPA1,TRPM2,TRPM8.Our products are only suitable for scientific research experiments, not for clinical experiments and human body.	price>
R-C-3251	AMG517 CAS:659730-32-2	AMG 517 is a potent and selective TRPV1 antagonist, and antagonizes capsaicin, proton, and heat activation of TRPV1.Our products are only suitable for scientific research experiments, not for clinical experiments and human body.	price>
R-C-3252	A-889425 CAS:1072921-02-8	A-889425 is a selective TRPV1 receptor antagonist.A-889425 blocks TRPV1 channels with an IC50 of 335nM(rat) and 34nM(human).Our products are only suitable for scientific research experiments, not for clinical experiments and human body.	price>
R-C-3253	MRS1477 CAS:212200-21-0	MRS1477 is a TRPV1 positive allosteric modulator.Our products are only suitable for scientific research experiments,not for clinical experiments and human body.	price>
R-C-3254	Mavatrep CAS:956274-94-5	Mavatrep is an orally bioavailable TRPV1 antagonist(Ki=6.5nM),exhibits minimal effect on the enzymatic activity(IC50>25μM)of CYP isoforms 3A4,1A2,and 2D6.Our products are only suitable for scientific research experiments, not for clinical experiments and human body.	price>
R-C-3255	A-1165442 CAS:1221443-94-2	A-1165442 is a potent,competitive and orally available TRPV1 antagonist with an IC50 of 9nM for human TRPV1. Our products are only suitable for scientific research experiments, not for clinical experiments and human body.	price>
R-C-3256	ORM-10962 CAS: 763926-98-3	ORM-10962 is a potent, highly selective sodium-calcium exchanger (NCX) inhibitor, with IC50 values of 67 and 55 nM for the reverse and forward mode inhibition, respectively. Our products are only suitable for scientific research experiments, not for clinical experiments and human body.	price>
R-C-3257	CGP 37157 CAS:75450-34-9	CGP-37157 is a potent,selective,and specific inhibitor of mitochondrial Na(+)-Ca2+ exchanger at concentrations≤10μM.Our products are only suitable for scientific research experiments, not for clinical experiments and human body.	price>
R-C-3258	ORM-10103 CAS:488847-28-5	ORM-10103 is a specific inhibitor of the Na+/Ca2+ exchanger(NCX),which decreases the NCX current with estimated IC50s of 55 and 67nM at -80 and at 20mV,respectively.Our products are only suitable for scientific research experiments, not for clinical experiments and human body.	price>

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