Catalog |
name |
Description |
price |
R-XASYS-00758 |
AZD8797,cas:911715-90-7 |
AZD8797 (C19H25N5OS2,403.56) is an allosteric non-competitive and orally active antagonist of the human CX3CR1 receptor; antagonizes CX3CR1 and CXCR2 with Kis of 3.9 and 2800 nM, respectively. |
price> |
R-XASYS-00759 |
Azelastine,cas:58581-89-8 |
Azelastine(C22H24ClN3O,381.90), an antihistamine, is a potent and selective histamine 1 (H1) antagonist. Azelastine can be used for the research of allergic rhinitis, asthma, diabetic hyperlipidemic and SARS-CoV-2. |
price> |
R-XASYS-00760 |
AZD3264,cas:1609281-86-8 |
AZD3264(C21H23N5O4S,441.5) is a selective IkB-kinase IKK2 inhibitor. |
price> |
R-XASYS-00761 |
AZD9496 maleate,cas:1639042-28-6 |
AZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). |
price> |
R-XASYS-00762 |
Azilsartan medoxomil monopotassium,cas:863031-24-7 |
Azilsartan medoxomil monopotassium(C30H23KN4O8,606.62) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. |
price> |
R-XASYS-00763 |
Azimilide,cas:149908-53-2 |
Azimilide(C23H28ClN5O3,457.95) is a class III antiarrhythmic compound, inhibits I(Ks) and I(Kr) in guinea-pig cardiac myocytes and I(Ks) (minK) channels expressed in Xenopus oocytes. |
price> |
R-XASYS-00764 |
AZM475271,cas:476159-98-5 |
AZM475271(C23H27ClN4O3,442.9) is a potent and selective Src kinase inhibitor with IC50 of 5 nM; no inhibitory activity on Flt3, KDR, Tie-2. |
price> |
R-XASYS-00765 |
Azt-pmap,cas:142629-81-0 |
Azt-pmap(C20H25N6O8P,508.42), a nucleoside analogue, is an aryl phosphate derivative of AZT. Azt-pmap shows anti-HIV activity. AZT is a nucleoside reverse transcriptase inhibitor (NRTI) for HIV infection. |
price> |
R-XASYS-00766 |
B-Raf IN 1,cas:950736-05-7 |
B-Raf IN 1(C29H24F3N5O,515.5) is a potent and selective B-Raf kinase inhibitor with an IC50 of 24 nM. |
price> |
R-XASYS-00767 |
B-Raf inhibitor 1 dihydrochloride,cas:1191385-19-9 |
B-Raf inhibitor 1 dihydrochloride(C26H21Cl3N8,551.86) is a potent Raf kinase inhibitor with Kis of 1 nM, 1 nM, and 0.3 nM for B-RafWT, B-RafV600E, and C-Raf, respectively. |
price> |