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Catalog	name	Description	price
R-C-2274	Cidofovir CAS: 113852-37-2	Cidofovir is an anti-CMV drug which can suppress CMV replication by selective inhibition of viral DNA polymerase and therefore prevention of viral replication and transcription.	price>
R-R-3974	(Rac)-Nebivolol CAS No.99200-09-6	(Rac)-Nebivolol ((Rac)-R 065824)/CAS No.99200-09-6 is a racemic isomer of Nebivolol. Nebivolol is a selective β1-adrenergic receptor antagonist with an IC50 value of 0.8 nM. Nebivolol can prevent up-regulation of Nox2/NADPH oxidase and lipoperoxidation in the early stages of ethanol-induced cardiac toxicity. Vasodilatory activity.	price>
R-C-2275	Cytarabine (U-19920A) CAS:147-94-4	Cytarabine(U-19920A,Cytarabin,Ara-C,Arabinofuranosyl Cytidine,Cytosine β-D-arabinofuranoside,Cytosine arabinoside,NSC 63878,NSC 287459)is an antimetabolic agent and DNA synthesis inhibitor with IC50 of 16 nM in wild-type CCRF-CEM cells.Cytarabine induces autophagy and apoptosis.	price>
R-R-3975	Terbutaline sulfate (Standard) CAS No.23031-32-5	Terbutaline (sulfate) (Standard)/CAS No.23031-32-5 is the analytical standard of Terbutaline (sulfate). This product is intended for research and analytical applications. Terbutaline sulfate is an orally active β2-adrenergic receptor agonist and an active metabolite of bambuterol. Terbutaline sulfate can be used in asthma symptom research.	price>
R-C-2276	Gemcitabine (LY-188011) CAS:95058-81-4	Gemcitabine(LY 188011)is a pyrimidine nucleoside analog antimetabolite and an antineoplastic agent.Gemcitabine inhibits DNA synthesis and repair,resulting in autophagyand apoptosis.	price>
R-R-3976	Isoxsuprine-d6 hydrochloride CAS No.2706004-35-3	Isoxsuprine-d6 (hydrochloride)/CAS No.2706004-35-3 is the deuterium labeled Isoxsuprine hydrochloride. Isoxsuprine hydrochloride is a beta-adrenergic receptor agonist with Kis of 13.65 μΜ and 3.48 μΜ for myometrial and placcntal beta-adrenergic receptor, respectively. Isoxsuprine hydrochloride is also a NMDA receptor antagonist.	price>
R-C-2277	Nelarabine CAS:121032-29-9	Nelarabine(Arranon,506U78)is a purine nucleoside analog and DNA synthesis inhibitor with IC50 from 0.067-2.15μM in tumor cells.	price>
R-R-3977	Azepexole dihydrochloride CAS No.36067-72-8	Azepexole (B-HT 933) dihydrochloride/CAS No.36067-72-8 is a potent and selective alpha 2-adrenoceptor agonist with pKis of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions (IC50= 78.72 nM).	price>
R-C-2278	Cladribine (RWJ 26251) CAS:4291-63-8	Cladribine(RWJ 26251,Leustatin,2-CdA,2-chlorodeoxyadenosine,2-Chloro-2-deoxyadenosine,CldAdo,Jk 6251,NSC 105014)is an adenosine deaminase inhibitor for U266,RPMI8226,and MM1.S cells with IC50 of approximately 2.43μM,0.75μM,and 0.18μM,respectively.	price>
R-R-3978	Betaxolol-d7 hydrochloride CAS No.1219802-92-2	Betaxolol-d7 (hydrochloride)/CAS No.1219802-92-2 is the deuterium labeled Betaxolol hydrochloride. Betaxolol Hydrochloride is a selective beta1 adrenergic receptor blocker that can be used for the research of hypertension and glaucoma.	price>
R-C-2279	Raltitrexed CAS:112887-68-0	Raltitrexed(Tomudex)is an inhibitor of thymidylate synthase and also is one of the strongest antimetabolites in use.	price>
R-R-3979	Cimbuterol CAS No.54239-39-3	Cimbuterol/CAS No.54239-39-3 is a β-adrenergic receptor agonist.	price>
R-C-2280	Clofarabine CAS:123318-82-1	Clofarabine is a second generation purine nucleoside analog with antineoplastic activity.Clofarabine is phosphorylated intracellularly to the cytotoxic active 5-triphosphate metabolite,which inhibits the enzymatic activities of ribonucleotide reductase and DNA polymerase,resulting in inhibition of DNA repair and synthesis of DNA and RNA.This nucleoside analog also disrupts mitochondrial function and membrane integrity,resulting in the release of pre-apoptotic factors,including cytochrome C and apoptotic-inducing factor,which activate apoptosis.	price>
R-R-3980	Tizanidine-d4 hydrochloride CAS No.1188263-51-5	Tizanidine-d4 (hydrochloride)/CAS No.1188263-51-5 is deuterium labeled Tizanidine (hydrochloride).	price>
R-C-2281	Go6976 CAS:136194-77-9	Go6976 is a potent PKC inhibitor with IC50 of 7.9nM,2.3nM,and 6.2nM for PKC(Rat brain),PKCα,and PKCβ1,respectively.Also a potent inhibitor of JAK2 and Flt3.	price>
R-R-3981	Guanfacine-13C,15N3 CAS No.1189924-28-4	Guanfacine-13C,15N3/CAS No.1189924-28-4 is the 13C and 15N labeled Guanfacine. Guanfacine is an orally active noradrenergic α2A agonist and has high selective for the α2A receptor subtype. Guanfacine has effects in producing hypotension and sedation.	price>
R-C-2282	Pomalidomide (CC-4047) CAS:19171-19-8	Pomalidomide,the third-generation immunomodulatory agent,acts as molecular glue. Pomalidomide interacts with the E3 ligase cereblon and induces degradation of essential Ikaros transcription factors.	price>
R-R-3982	Talibegron hydrochloride CAS No.178600-17-4	Talibegron hydrochloride (ZD2079 hydrochloride)/CAS No.178600-17-4 is a potent β3-adrenoceptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Talibegron hydrochloride has potent vasorelaxant effect.	price>
R-C-2283	CC-90009 CAS:1860875-51-9	CC-90009 is a cereblon modulator.CC-90009 specifically binds to CRBN,thereby affecting the activity of the ubiquitin E3 ligase complex.This leads to the ubiquitination of certain substrate proteins and induces the proteasome-mediated degradation of certain transcription factors,including Ikaros(IKZF1)and Aiolos (IKZF3),which are transcriptional repressors in T-cells.This reduces the levels of these transcription factors,and modulates the activity of the immune system, which may include the activation of T-lymphocytes.	price>
R-R-3983	Perphenazine-d8 dihydrochloride CAS No.2070015-23-3	Perphenazine-d8 (dihydrochloride)/CAS No.2070015-23-3 is the deuterium labeled Perphenazine, which is a typical antipsychotic agent(5-HT, Dopamine receptor ligand).	price>

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