Indophagolin CAS No.1207660-00-1
Indophagolin CAS No.1207660-00-1
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-2121 | 5mg | 280.00 | + Add to cart |
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R-R-2121 | 10mg | 460.00 | + Add to cart |
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Product description
Indophagolin/CAS No.1207660-00-1 is a potent, indoline-containing autophagy inhibitor (IC50=140 nM). Indophagolin antagonizes the purinergic receptor P2X4 as well as P2X1 and P2X3 with IC50s of 2.71, 2.40 and 3.49 μM, respectively. Indophagolin also antagonizes the Gq-protein-coupled P2Y4, P2Y6, and P2Y11 receptors (IC50s =3.4~15.4 μM). Indophagolin has a strong antagonistic effect on serotonin receptor 5-HT6 (IC50=1.0 μM) and a moderate effect on receptors 5-HT1B, 5-HT2B, 5-HT4e, and 5-HT7.
Appearance | N/A |
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Molecular Weight | 523.75 |
Purity | >90% |
CAS | 1207660-00-1 |
Formula | C19H15BrClF3N2O3S |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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