GNE-781 CAS No.1936422-33-1
GNE-781 CAS No.1936422-33-1
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-2445 | 5mg | 360.00 | + Add to cart |
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R-R-2445 | 10mg | 610.00 | + Add to cart |
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Product description
GNE-781/CAS No.1936422-33-1 is an orally active, highly potent and selective CBP inhibitor with an IC50 of 0.94 nM in TR-FRET assay. GNE-781 also inhibits BRET and BRD4(1) with IC50s of 6.2 nM and 5100 nM, respectively. GNE-781 displays antitumor activity in an MOLM-16 AML xenograft model.
Appearance | N/A |
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Molecular Weight | 525.59 |
Purity | >90% |
CAS | 1936422-33-1 |
Formula | C27H33F2N7O2 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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