GSK778 CAS No.2451862-42-1
GSK778 CAS No.2451862-42-1
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-2446 | 5mg | 380.00 | + Add to cart |
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R-R-2446 | 10mg | 630.00 | + Add to cart |
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Product description
GSK778 (iBET-BD1)/CAS No.2451862-42-1 is a potent and selective BD1 bromodomain inhibitor of the BET proteins, with IC50s of 75 nM (BRD2 BD1), 41 nM (BRD3 BD1), 41 nM (BRD4 BD1), and 143 nM (BRDT BD1), respectively. GSK778 phenocopies the effects of pan-BET inhibitors in cancer models.
Appearance | N/A |
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Molecular Weight | 511.61 |
Purity | >90% |
CAS | 2451862-42-1 |
Formula | C30H33N5O3 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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