Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-2887	KH7 CAS No.330676-02-3	KH7/CAS No.330676-02-3 is a specific double adenyl cyclone (sAC) inhibitor, with IC50s of 3-10 μM toward both purified human sACT recombinant proteins and highly expressed sACT terolog in cellular assays KH7 is also a cAMP inhibitor	price>
R-R-2888	LRE1 CAS No.1252362-53-0	LRE1/CAS No.1252362-53-0 is a specific and allosteric inhibitor of soluble adenylyl cyclase.	price>
R-R-2889	TDI-10229 CAS No.2810887-45-5	TDI-10229/CAS No.2810887-45-5 is a potent and orally bioavailable inhibitor of soluble adenylyl cyclase (sAC, ADCY10). TDI-10229 displays nanomolar inhibition of sAC in both biochemical and cellular assays (IC50 of 195 nM) and exhibits mouse pharmacokinetic properties sufficient to warrant its use as an in vivo tool compound.	price>
R-R-2890	Fipexide CAS No.34161-24-5	Fipexide/CAS No.34161-24-5, a parachloro-phenossiacetic acid derivative, is an orally active nootropic agent. Fipexide reduces striatal adenylate cyclase activity. Fipexide has positive effect on cognitive performance by dopaminergic neurotransmission. Fipexide is used for senile dementia research. Fipexide acts as a chemical inducer in callus formation, shoot regeneration and Agrobacterium infection.	price>
R-R-2891	SKF-83566 CAS No.99295-33-7	SKF-83566/CAS No.99295-33-7 is a potent, blood-brain permeable and orally active D1-like dopamine receptor (D1DR) antagonist and a weaker competitive antagonist at the vascular 5-HT2 receptor (Ki=11 nM). SKF-83566 is a competitive DAT (dopamine transporter) inhibitor with an IC50 of 5.7 μM. SKF-83566 also shows selective inhibition for adenylyl cyclase 2 (AC2) over AC1 and AC5 in the isolated rabbit thoracic aorta.	price>
R-R-2892	ST034307 CAS No.133406-29-8	ST034307/CAS No.133406-29-8 is a potent and selective adenylyl cyclase 1 (AC1) inhibitor, with IC50 of 2.3 μM.	price>
R-R-2893	NKY80 CAS No.299442-43-6	NKY80/CAS No.299442-43-6 is a potent, selective and non-competitive adenylyl cyclase (AC) type V isoform inhibitor with IC50s of 8.3 µM, 132 µM and 1.7 mM for type V, III and II, respectively. NKY80 is a non-nucleoside quinazolinone and regulates the AC catalytic activity in heart and lung tissues.	price>
R-C-1194	LY310762 CAS:192927-92-7	LY310762 is a 5-HT1D antagonist with Ki of 249 nM, having a weaker affinity for 5-HT1B receptor.	price>
R-R-2894	Guanylyl imidodiphosphate lithium CAS No.64564-03-0	Guanylyl imidodiphosphate (Gpp(NH)p) lithium/CAS No.64564-03-0, a non-hydrolyzable GTP analogue, increases adenylate cyclase activity.	price>
R-R-2895	TDI-11861 CAS No.2857049-72-8	TDI-11861/CAS No.2857049-72-8 is second-generation soluble Adenylyl Cyclase (sAC, ADCY10) inhibitor with slow dissociation rates. TDI-11861 inhibits sAC cellular with an IC50 value of 5.5 nM.	price>

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