Product apis-gpcr-g-protein

Home > products > apis> gpcr-g-protein

Catalog	name	Description	price
R-R-2860	GCGR antagonist 2 CAS No.280134-25-0	GCGR antagonist 2/CAS No.280134-25-0, a Furan-2-carbohydrazide, is an orally active glucagon receptor antagonist. GCGR antagonist 2 binds to hGluR with an Kd value of 2.3 nM, and inhibits rat receptor with an IC50 value of 0.43 nM. GCGR antagonist 2 inhibits glucagon-stimulated glycogenolysis.	price>
R-R-2861	Exendin-3/4 (59-86) CAS No.1263874-37-8	Exendin-3/4 (59-86)/CAS No.1263874-37-8 is a Exendin-4 peptide derivative.	price>
R-R-2862	{Val1}-Exendin-3/4	{Val1}-Exendin-3/4 is the first N-terminal 1-28 residues of Exendin-4 peptide.	price>
R-C-1163	OPC 21268 CAS:131631-89-5	OPC21268 is a non-peptide AVP Receptor V(Vasopressin Receptor)antagonist that shows 1000-fold selectivity for V1 receptors over V2 receptors.	price>
R-R-2864	GLP-1 (1-36) amide (human, rat) (TFA)	GLP-1 (1-36) amide (human, rat) (Glucagon-like Peptide 1 (1-36) amide (human, rat) ) TFA is a molecular variant of glucagon-like peptide 1 (GLP-1)-(7-36) amide. GLP-1 (1-36) amide (human, rat) TFA can stimulate [14C]aminopyrine accumulation on enzymatically dispersed enriched rat parietal cells.	price>
R-R-2865	SAR441255 TFA	SAR441255 TFA is a potent unimolecular peptide GLP-1/GIP/GCG receptor triagonist. SAR441255 TFA displays high potency with balanced activation of all three target receptors.?SAR441255 TFA shows positive acute glucoregulatory effectss in diabetic obese monkeys.	price>
R-R-2866	V-0219 CAS No.878453-71-5	V-0219 (Compound 9)/CAS No.878453-71-5 is an orally active, positive allosteric modulator (PAM) of the glucagon-like peptide-1 receptor (GLP-1R). V-0219 can be used for obesity-associated diabetes research.	price>
R-R-2867	V-0219 hydrochloride CAS No.2922283-73-4	V-0219 hydrochloride (Compound 9)/CAS No.2922283-73-4 is an orally active, positive allosteric modulator (PAM) of the glucagon-like peptide-1 receptor (GLP-1R). V-0219 hydrochloride can be used for obesity-associated diabetes research.	price>
R-R-2868	Apraglutide TFA	Apraglutide TFA (FE 203799 TFA), a synthetic 33-amino-acid peptide and a long-acting GLP-2 analogue, enhances adaptation and linear intestinal growth in a neonatal piglet model of short bowel syndrome with total resection of the ileum.	price>
R-C-1169	GW 627368 CAS： 439288-66-1	GW627368(GW627368X)is a novel,potent and selective competitive antagonist of prostanoid EP4 receptor with additional human TP receptor affinity, with pKi values of 7.0 and 6.8 for human prostanoid EP4 and TP receptors respectively.	price>

...

163