Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-2858	GLP-1R agonist 3 CAS No.2428640-18-8	GLP-1R agonist 3/CAS No.2428640-18-8 is a potent agonist of GLP-1R. GLP-1R agonist 3 is a thickened imidazole derivative compound. Glucagon-like peptide-1 (GLP-1) is an intestinal hypoglycemic hormone secreted by L-cells in the lower gastrointestinal tract. GLP-1R agonist 3 has the potential for the research of diabetes (extracted from patent WO2021197464A1, compound 1).	price>
R-R-2859	Glucagon receptor antagonists-1 CAS No.503559-84-0	Glucagon receptor antagonists-1/CAS No.503559-84-0 is a highly potent glucagon receptor antagonist.	price>
R-R-2860	GCGR antagonist 2 CAS No.280134-25-0	GCGR antagonist 2/CAS No.280134-25-0, a Furan-2-carbohydrazide, is an orally active glucagon receptor antagonist. GCGR antagonist 2 binds to hGluR with an Kd value of 2.3 nM, and inhibits rat receptor with an IC50 value of 0.43 nM. GCGR antagonist 2 inhibits glucagon-stimulated glycogenolysis.	price>
R-R-2861	Exendin-3/4 (59-86) CAS No.1263874-37-8	Exendin-3/4 (59-86)/CAS No.1263874-37-8 is a Exendin-4 peptide derivative.	price>
R-R-2862	{Val1}-Exendin-3/4	{Val1}-Exendin-3/4 is the first N-terminal 1-28 residues of Exendin-4 peptide.	price>
R-C-1163	OPC 21268 CAS:131631-89-5	OPC21268 is a non-peptide AVP Receptor V(Vasopressin Receptor)antagonist that shows 1000-fold selectivity for V1 receptors over V2 receptors.	price>
R-R-2863	Tirzepatide CAS No.2023788-19-2	Tirzepatide (LY3298176)/CAS No.2023788-19-2 is a glucose-dependent insulin nutritive polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor dual agonist. Tirzepatide has neuroprotective effects and can be used in the study of type 2 diabetes, diabetes-related neuropathy and obesity.	price>
R-R-2864	GLP-1 (1-36) amide (human, rat) (TFA)	GLP-1 (1-36) amide (human, rat) (Glucagon-like Peptide 1 (1-36) amide (human, rat) ) TFA is a molecular variant of glucagon-like peptide 1 (GLP-1)-(7-36) amide. GLP-1 (1-36) amide (human, rat) TFA can stimulate [14C]aminopyrine accumulation on enzymatically dispersed enriched rat parietal cells.	price>
R-R-2865	SAR441255 TFA	SAR441255 TFA is a potent unimolecular peptide GLP-1/GIP/GCG receptor triagonist. SAR441255 TFA displays high potency with balanced activation of all three target receptors.?SAR441255 TFA shows positive acute glucoregulatory effectss in diabetic obese monkeys.	price>
R-R-2866	V-0219 CAS No.878453-71-5	V-0219 (Compound 9)/CAS No.878453-71-5 is an orally active, positive allosteric modulator (PAM) of the glucagon-like peptide-1 receptor (GLP-1R). V-0219 can be used for obesity-associated diabetes research.	price>

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