Product apis-gpcr-g-protein

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Catalog	name	Description	price
R-R-2832	Glucagon receptor antagonists-3 CAS No.202917-17-7	Glucagon receptor antagonists-3/CAS No.202917-17-7 is a highly potent glucagon receptor antagonist.	price>
R-R-2833	Mazdutide CAS No.2259884-03-0	Mazdutide (IBI-362; LY-3305677)/CAS No.2259884-03-0 is a long-acting synthetic oxyntomodulin analog. Mazdutide is also a co-agonist of glucagon-like peptide (GLP-1R) and?glucagon receptor?(GCGR). Mazdutide binds human and mouse?GCGR?(Ki: 17.7 nM and 15.9 nM, respectively) and GLP-1R (Ki: 28.6 nM and 25.1 nM, respectively) and stimulates?insulin?secretion from mouse islets (EC50: 5.2 nM). Mazdutide is used in studies of obesity and type 2 diabetes (T2D).	price>
R-R-2834	L-168049 CAS No.191034-25-0	L-168049/CAS No.191034-25-0 is a potent, selective, orally active and non-competitive glucagon receptor antagonist with IC50s of 3.7 nM, 63 nM, and 60 nM for human, murine, and canine glucagon receptors, respectively.	price>
R-R-2835	Shanzhiside methyl ester CAS No.64421-28-9	Shanzhiside methy lester/CAS No.64421-28-9 is isolated from lamiophlomis rotata. Shanzhiside methyl ester is a small molecule glucagon-like peptide-1 (GLP-1) receptor agonist and has the ability to induce anti-allodynic tolerance.	price>
R-R-2836	VU0453379 hydrochloride	VU0453379 hydrochloride is a highly selective and central nervous system (CNS) penetrant positive allosteric modulator (PAM) of glucagon-like peptide-1R (GLP-1R) with an EC50 of 1.3 μM.	price>
R-R-2837	GLP-1(7-36), amide TFA	GLP-1(7-36), amide TFA is a major intestinal hormone that stimulates glucose-induced insulin secretion from β cells.	price>
R-R-2838	Dapiglutide CAS No.2296814-85-0	Dapiglutide (ZP7570)/CAS No.2296814-85-0 is a long-acting glucagon-like peptide-1 receptor 1R (GLP-1R)/Glucagon-like peptide-2 receptor (GLP-2R) dual agonist. Dapiglutide can be used for short bowel syndrome (SBS) research.	price>
R-R-2839	Taspoglutide CAS No.275371-94-3	Taspoglutide/CAS No.275371-94-3 is a long-acting glucagon-like peptide 1 (GLP-1) receptor agonist developed for treatment of type 2 diabetes, with an EC50 value of 0.06 nM.	price>
R-R-2840	Glucagon receptor antagonists-2 CAS No.202917-18-8	Glucagon receptor antagonists-2/CAS No.202917-18-8 is a highly potent glucagon receptor antagonist.	price>
R-R-2841	GLP-1R modulator L7-028 CAS No.2648317-95-5	GLP-1R modulator L7-028/CAS No.2648317-95-5 is an allosteric modulator enhancing GLP-1 binding to GLP-1R via a transmembrane site (EC50 11.01 ± 2.73 μM).	price>

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