Catalog name Description price
R-C-3161 SR-12813 CAS:126411-39-0 SR-12813 is a pregnane X receptor(PXR)agonist and HMG-CoA reductase inhibitor with an IC50 of 850 nM. price>
R-C-3162 Epristeride CAS:119169-78-7 Epristeride is a selective and specific uncompetitive inhibitor of human steroid 5 alpha-reductase isoform 2. price>
R-C-3163 AR-231453 CAS:733750-99-7 AR-231453 is a potent and selective small molecule agonis of GPR119 that enhances glucose dependent insulin secretion and glucagon like peptide-1 (GLP-1) release. price>
R-C-3164 6-OAU CAS:83797-69-7 6-OAU (GTPL5846, 6-n-octylaminouracil) is a surrogate agonist of G protein-coupled receptor 84 (GPR84) that activates human GPR84 in the presence of Gqi5 chimera in HEK293 cells with EC50 of 105 nM in the PI assay.6-OAU(GTPL5846,6-n-octylaminouracil)increases [35S]GTPγS incorporated in Sf9 cell membranes expressing human GPR84-Gαi fusion protein with EC50 of 512nM. price>
R-C-3165 Versipelostatin Versipelostatin is a novel GRP78/Bip molecular chaperone down-regulator of microbial origin that was isolated from the metabolite of Streptomyces versipellis strain 4083-SVS6.Our products are only suitable for scientific research experiments, not for clinical experiments and human body. price>
R-C-3167 NCRW0005-F05 CAS:342779-66-2 NCRW0005-F05, first antagonist selective for GPR139 (IC50 value 0.21 uM); a useful tool to study GPR139 pharmacology, especially in combination with the GPR139 agonist JNJ 63533054.Our products are only suitable for scientific research experiments, not for clinical experiments and human body. price>
R-C-3168 BMS-564929 CAS:627530-84-1 BMS-564929 is a novel, highly potent, orally active, nonsteroidal tissue selective androgen receptor (AR) modulator, and this compound has been advanced to clinical trials for the treatment of age-related functional decline. Our products are only suitable for scientific research experiments, not for clinical experiments and human body. price>
R-C-3169 AZD3514 CAS:1240299-33-5 AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2M and has ability of reducing AR protein expression.Our products are only suitable for scientific research experiments, not for clinical experiments and human body. price>
R-C-3170 GSK-2881078 CAS :1539314-06-1 GSK 2881078 is a nonsteroidal selective modulator of androgen receptor that is potentially used for the treatment of cachexia.Our products are only suitable for scientific research experiments, not for clinical experiments and human body. price>
R-C-3171 MK-0773 CAS: 606101-58-0 MK-0773,one of selective androgen receptor modulators(SARMs),is a 4-aza-steroid that exhibited tissue selectivity in humans (IC50=6.6nM).Our products are only suitable for scientific research experiments, not for clinical experiments and human body. price>