Catalog |
name |
Description |
price |
R-XASYS-00617 |
Afegostat D-Tartrate,cas:957230-65-8 |
Afegostat D-Tartrate(C10H19NO9,297.3) is a pharmacological chaperone, which specifically and reversibly binds acid-β-glucosidase (GCase) in the endoplasmic reticulum (ER) with high affinity. |
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R-XASYS-00618 |
AFN-1252,cas:620175-39-5 |
AFN-1252(Debio 1452)(C22H21N3O3,375.4) is a potent inhibitor of enoyl-acyl carrier protein reductase (FabI), inhibited all clinical isolates of Staphylococcus aureus and Staphylococcus epidermidis at concentrations of≤0.12μg/ml. |
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R-XASYS-00619 |
AG3340 hydrochloride,cas:1435779-45-5 |
Prinomastat hydrochloride (AG3340 hydrochloride)(C18H22ClN3O5S2,459.97) is a broad spectrum, potent, orally active metalloproteinase (MMP) inhibitor with IC50s of 79, 6.3 and 5.0 nM for MMP-1, MMP-3 and MMP-9, respectively. Prinomastat hydrochloride inhibits MMP-2, MMP-3 and MMP-9 with Kis of 0.05 nM, 0.3 nM and 0.26 nM, respectively. Prinomastat hydrochloride can cross blood-brain barrier. Antitumor avtivity. |
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R-XASYS-00620 |
Agarotetrol,cas:69809-22-9 |
Agarotetrol(C17H18O6,318.3) is a chromone derivative originally isolated from agarwood, a component of incense and traditional medicines. |
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R-XASYS-00621 |
Agerafenib hydrochloride,cas:1227678-26-3 |
Agerafenib hydrochloride(C24H23ClF3N5O5,553.92) is a highly potent and orally efficacious inhibitor of BRAFV600E with a Kd of 14 nM. |
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R-XASYS-00622 |
AGI-24512,cas:2201066-53-5 |
AGI-24512(C24H24N4O2,400.48) is a potent methionine adenosyltransferase 2α (MAT2A) inhibitor, with an IC50 of 8 nM. AGI-24512 triggers DNA damage response. AGI-24512 can block proliferation of MTAP-deleted cancer cells in vitro. AGI-24512 can be used for researching anticancer. |
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R-XASYS-00623 |
AGL-2263,cas:638213-98-6 |
AGL 2263(C17H10N2O5,322.3) is an inhibitor of the insulin-like growth factor 1 receptor (IGF-1R; IC50 = 0.43μM).It also inhibits the insulin receptor (IR), protein kinase B (PKB), and Src in a cell-free assay (IC50s = 0.4,55, and 2.2μM respectively). |
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R-XASYS-00624 |
Aglafoline,cas:143901-35-3 |
Aglafoline(C28H28O8,492.52) inhibits in a selective and concentration-dependent manner the aggregation and ATP release reaction induced in washed rabbit platelets by PAF (platelet-activating factor). |
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R-XASYS-00625 |
AGN 193109,cas:171746-21-7 |
AGN 193109 (GMP)(C28H24O2,392.49) is AGN 193109 (HY-U00449) produced by using GMP guidelines. GMP small molecules works appropriately as an auxiliary reagent for cell therapy manufacture. AGN 193109 is a specific and highly effective retinoic acid receptor (RAR) antagonist. |
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R-XASYS-00626 |
AH 6809,cas:33458-93-4 |
AH 6809(C17H14O5,298.3) is an antagonist of EP and DP receptor, with Kis of 1217, 1150, 1597, and 1415 nM for the cloned human EP1, EP2, EP3-III, and DP receptor respectively. AH 6809 has a Ki of 350 nM for mouse EP2 receptor. |
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