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Catalog	name	Description	price
R-R-4378	SKF-75670 hydrobromide CAS No.62717-63-9	SKF-75670 hydrochloride/CAS No.62717-63-9 is a Dopamine D1 receptor partial agonist. SKF-75670 hydrochloride is also a Cocaine antagonist.	price>
R-C-2679	Carmofur CAS：61422-45-5	Carmofur(HCFU),a derivative of 5-Fluorouracil,is an antineoplastic agent.Carmofur is an inhibitor of acid ceramidase with an IC50 of 79nM for the rat enzyme.Carmofur inhibits the SARS-CoV-2 main protease(Mpro).Carmofur Inhibits SARS-CoV-2 in Vero E6 cell with an EC50 of 24.3μM.	price>
R-R-4379	Bromopride CAS No.4093-35-0	Bromopride/CAS No.4093-35-0 is a dopamine antagonist with prokinetic properties, widely used as an antiemetic.	price>
R-C-2680	Altretamine CAS：645-05-6	Altretamine is classified as an alkylating antineoplastic agent.This unique structure is believed to damage tumor cells through the production of the weakly alkylating species formaldehyde,a product of CYP450-mediated N-demethylation.	price>
R-R-4380	Ziprasidone amino acid CAS No.1159977-64-6	Ziprasidone amino acid (Ziprasidone Impurity C)/CAS No.1159977-64-6 is an impurity of Ziprasidone. Ziprasidone is a combined 5-HT (serotonin) and dopamine receptor antagonist. Ziprasidone exhibits potent effects of antipsychotic activity .	price>
R-C-2681	Amonafide CAS： 69408-81-7	Amonafide is a topoisomerase II inhibitor and DNA intercalator that induces apoptotic signaling by blocking the binding of Topo II to DNA.	price>
R-R-4381	ST-836 hydrochloride CAS No.1415564-68-9	ST-836 hydrochloride (compound 34)/CAS No.1415564-68-9 is a potent dopamine receptor ligand with Ki values of 4.5 nM, 132 nM for D3 and D2, respectively. ST-836 hydrochloride has the potential for Parkinson disease.	price>
R-C-2682	CRT0044876 CAS：6960-45-8	CRT0044876 is a potent BER inhibitor or DNA Base Excision Repair Pathway Inhibitor (APE1 IC50-3 microM).CRT0044876 potentiates the cytotoxicity of several DNA base-targeting compounds,with accumulation of apurinic sites.	price>
R-R-4382	CGP 25454A CAS No.104391-26-6	CGP 25454A/CAS No.104391-26-6 is a selective presynaptic dopamine autoreceptor antagonist which induces the increase of dopamine and acetyl choline. CGP 25454A can be used for major depression research.	price>
R-C-2683	Leflunomide CAS:75706-12-6	Leflunomide(HWA486,RS-34821,SU101,Arava)is a pyrimidine synthesis and protein tyrosine kinase inhibitor belonging to the DMARD,used as an immunosuppressant agent.The active metabolite of Leflunomide is A77 1726,which inhibits dihydroorotate dehydrogenase (DHODH).Leflunomide is also an agonist of the AhR.	price>
R-R-4383	Zuclopenthixol-d4 succinate CAS No.1246833-97-5	Zuclopenthixol-d4 (succinate)/CAS No.1246833-97-5 is the deuterium labeled Zuclopenthixol. Zuclopenthixol is a thioxanthene derivative which acts as a mixed dopamine D1/D2 receptor antagonist.	price>
R-C-2684	RX-3117 CAS：865838-26-2	RX-3117(TV-1360;Fluorocyclopentenylcytosine)is novel a cytidine analog;shows anticancer activity in several cancer cell lines,including gemcitabine-resistant variants.	price>
R-R-4384	L-DOPA-2,5,6-d3 CAS No.53587-29-4	L-DOPA-2,5,6-d3/CAS No.53587-29-4 is the deuterium labeled L-DOPA. L-DOPA (Levodopa) is an orally active metabolic precursor of neurotransmitters dopamine. L-DOPA can cross the blood-brain barrier and is converted into dopamine in the brain.	price>
R-C-2685	LY2334737 CAS：892128-60-8	LY2334737 is an nucleoside analog and is an orally active prodrug of Gemcitabine.LY2334737 exhibits inhibitory activity against enterovirus A71(EV-A71)infection.LY2334737 has antiviral and anticancer effects.	price>
R-R-4385	Propionylpromazine-d6 hydrochloride CAS No.1262770-67-1	Propionylpromazine-d6 (hydrochloride)/CAS No.1262770-67-1 is the deuterium labeled Propionylpromazine hydrochloride. Propionylpromazine hydrochloride (Propiopromazine hydrochloride), a dopamine receptor D2 (DRD2) antagonist, can be used in the research of Parkinson disease.	price>
R-C-2686	Evofosfamide (TH-302) CAS：918633-87-1	Evofosfamide(TH-302)is a hypoxia-activated prodrug with IC50 of 10μM and 1000 μM in hypoxia(N2)and normoxia(21% O2),respectively.	price>
R-R-4386	PD 168568 dihydrochloride CAS No.1782532-06-2	PD 168568 dihydrochloride/CAS No.1782532-06-2 is a orally active and potent dopamine receptor D4 (DRD4) antagonist. PD 168568 dihydrochloride contains an isoindolinone and is selective for the D4 receptor versus D2 and D3, with Ki values of 8.8, 1842, and 2682 nM, respectively. PD 168568 dihydrochloride can be used for glioblastoma (GBM) research.	price>
R-R-4387	Amisulpride-d5 CAS No.1216626-17-3	Amisulpride-d5/CAS No.1216626-17-3 is the deuterium labeled Amisulpride. Amisulpride is a dopamine D2/D3 receptor antagonist with Kis of 2.8 and 3.2 nM for human dopamine D2 and D3, respectively.	price>
R-R-4388	Cabergoline-d5 CAS No.1426173-20-7	Cabergoline-d5/CAS No.1426173-20-7 is the deuterium labeled Cabergoline. Cabergoline is an ergot derived-dopamine D2-like receptor agonist that has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respectively).	price>
R-C-2689	Calyculin A CAS：101932-71-2	Calyculin A is a natural,cell-permeable inhibitor of the serine-threonine protein phosphatases(PP)PP1 and PP2A(IC50s=0.3-0.7 and 0.5-1nM,respectively).It is without significant effect against PP2B,PP2C,and PP4.2 Through its effects on PP1 and PP2A,calyculin A has been shown to either promote or inhibit cancer cell growth in tumor cell lines and animal models.	price>

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