Xi'an ruixi Biological Technology Co

Home > Keywords >

Catalog	name	Description	price
R-R-4307	Lisuride maleate CAS No.19875-60-6	Lisuride (maleate)/CAS No.19875-60-6 is a potent agonist of dopamine with a probably direct action on dopaminergic receptors. Lisuride (maleate) is an ergot derivative. Lisuride (maleate) releases the premenstrual mastalgia without significant side effects.	price>
R-C-2608	Necrostatin 2 CAS:852391-19-6	Necrostatin 2(Nec-2)is a novel and potent necroptosis inhibitor with EC50 of 50 nM.It is an analog of necrostatin 1(nec-1).Necroptosis is a mechanism of necrotic cell death induced by apoptotic stimuli in the form of death domain receptor engagement by their respective ligands under conditions where apoptotic execution is prevented.	price>
R-R-4308	L-741626 CAS No.81226-60-0	L-741626/CAS No.81226-60-0 is a selective D2 dopamine receptor antagonist, with the Ki values of 2.4, 100 and 220 nM for human D2, D3 and D4 receptors respectively.	price>
R-C-2609	TLQP 21 CAS:869988-94-3	TLQP-21,a VGF-derived peptide endowed of endocrine and extraendocrine properties,is a potent G-protein-coupled receptor complement-3a receptor 1(C3aR1)agonist(EC50:mouse TLQP-21=10.3μM;human TLQP-21=68.8μM).TLQP-21 activates C3aR1 to induce an increase of intracellular Ca2+.TLQP-21 is used for the research in regulation of nociception and other relevant physiologic functions.	price>
R-R-4309	3-O-Methyldopa CAS No.300-48-1	3-O-Methyldopa (3-Methoxy-L-tyrosine)/CAS No.300-48-1 is a metabolite of L-DOPA which is formed by catechol-O-methyltransferase (COMT). 3-O-Methyldopa competitively inhibits the pharmacodynamics of l-DOPA and dopamine.	price>
R-C-2610	YM155 (Sepantronium Bromide) CAS:781661-94-7	YM155(Sepantronium Bromide)is a potent survivin suppressant by inhibiting Survivin promoter activity with IC50 of 0.54nM in HeLa-SURP-luc and CHO-SV40-luc cells;does not significantly inhibit SV40 promoter activity,but is observed to slightly inhibit the interaction of Survivin with XIAP.	price>
R-R-4310	Droperidol CAS No.548-73-2	Droperidol/CAS No.548-73-2 is a butyrophenone-type Dopamine-2 receptor antagonist.	price>
R-C-2611	SC-10 CAS:102649-79-6	SC-10 is a PKC activator.It acts by stimulating PKC mediated myosin light chain phosphorylation without activating MLC kinase.	price>
R-R-4311	Loxapine succinate CAS No.27833-64-3	Loxapine succinate/CAS No.27833-64-3 is an orally active dopamine inhibitor, 5-HT receptor antagonist and also a dibenzoxazepine anti-psychotic agent. Loxapine can also suppresses bacterial efflux pump activity and inhibit intracellular multiple-antibiotic-resistant Salmonella enterica serovar Typhimurium in macrophages.	price>
R-C-2612	ML347 CAS:1062368-49-3	ML347(DN193719)is a highly selective ALK1/ALK2 inhibitor with IC50s of 46/32nM; shows>300-fold selectivity for ALK2 vs.	price>
R-R-4312	Nomifensine CAS No.24526-64-5	Nomifensine/CAS No.24526-64-5 is a norepinephrine-dopamine reuptake inhibitor, increases the amount of synaptic norepinephrine and dopamine available to receptors by blocking the dopamine and norepinephrine reuptake transporters.	price>
R-C-2613	SR-3677 CAS:1072959-67-1	SR-3677 is a novel,potent and highly selective inhibitor of Rho Kinase(ROCK-II) with the IC50 value of ~0.3nM in enzyme and cell based assays.	price>
R-R-4313	A68930 hydrochloride CAS No.130465-39-3	A68930 hydrochloride/CAS No.130465-39-3, as a dopamine D1 receptor agonist, can be used for the research of bronchiectasis.	price>
R-C-2614	DMH-1 CAS:1206711-16-1	DMH-1 is a potent and selective BMP inhibitor with IC50s of 27/107.9/<5/47.6 nM for ALK1/ALK2/ALK3/ALK6,respectively.	price>
R-R-4314	Amisulpride CAS No.71675-85-9	Amisulpride/CAS No.71675-85-9 is a dopamine D2/D3 receptor antagonist with Kis of 2.8 and 3.2 nM for human dopamine D2 and D3, respectively.	price>
R-C-2615	Midostaurin (PKC412) CAS:120685-11-2	Midostaurin(PKC412;CGP 41251)is a multi-targeted protein kinase inhibitor which inhibits PKCα/β/γ,Syk,Flk-1,Akt,PKA,c-Kit,c-Fgr,c-Src,FLT3,PDFRβ and VEGFR1/2 with IC50s ranging from 22-500nM.	price>
R-R-4315	Clebopride malate CAS No.57645-91-7	Clebopride malate/CAS No.57645-91-7 is a dopamine antagonist drug with antiemetic and prokinetic properties used to treat functional gastrointestinal disorders.	price>
R-C-2616	Calphostin C CAS:121263-19-2	The calphostins are a class of closely related chemical compounds isolated from the fungus Cladosporium cladosporioides.The known calphostins include calphostin A,calphostin B,calphostin C,calphostin D,and calphostin I.The calphostins are inhibitors of protein kinase C(PKC).	price>
R-R-4316	Nomifensine maleate CAS No.32795-47-4	Nomifensine maleate/CAS No.32795-47-4 is a selective inhibitor of dopamine uptake, used in adult attention deficit disorder.	price>
R-C-2617	PKC fragment (530-558)	Potent activator of protein kinase C(Ka~10 mM);corresponds to residues 530-558 of the catalytic domain of PKC.	price>

636637638639640641 642643644645646