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Catalog	name	Description	price
R-R-4122	Arvanil CAS No.128007-31-8	Arvanil/CAS No.128007-31-8 is a ligand for vanilloid receptor 1 (VR1) and cannabinoid 1 (CB1). Arvanil can inhibit spasticity, as a potent neuroprotectant.	price>
R-C-2423	Myosmine CAS:532-12-7	Myosmine is not only one of the minor tobacco alkaloids but is also present in various foods.Myosmine has low affinity against a4b2 nicotinic acetylcholinergic receptors(nAChR)with Ki of 3300nM.	price>
R-R-4123	Taranabant ((1R,2R)stereoisomer) CAS No.701977-08-4	Taranabant (1R,2R)stereoisomer/CAS No.701977-08-4 is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist.	price>
R-C-2424	Amfebutamone (Bupropion) HCl CAS:31677-93-7	Amfebutamone(Bupropion)HCl is a selective norepinephrine-dopamine reuptake inhibitor with IC50 of 6.5 and 3.4uM for the reuptake of dopamine and norepinephrine,respectively.	price>
R-R-4124	Drinabant CAS No.358970-97-5	Drinabant (AVE1625)/CAS No.358970-97-5 is an orally active CB1 receptor antagonist. Drinabant (AVE1625) inhibits the agonist-stimulated calcium signal with IC50 values of 25 nM and 10 nM for the hCB1-R and rCB1-R, respectively, and is ineffective for the hCB2-R.	price>
R-C-2425	Galanthamine HBr CAS:1953-04-4	Galantamine Hydrobromide is the hydrobromide salt form of galantamine,a tertiary alkaloid with anticholinesterase and neurocognitive-enhancing activities.It is an alkaloid acetylcholinesterase inhibitor.Galantamine competitively and reversibly inhibits acetylcholinesterase,thereby increasing the concentration and enhancing the action of acetylcholine(Ach).	price>
R-R-4125	CB65 CAS No.913534-05-1	CB65/CAS No.913534-05-1 is a potent and high affinity CB2 selective agonist with a Ki value of 3.3 nM. CB65 exhibits a Ki of >1000 nM for CB1 receptor.	price>
R-C-2426	Rocuronium Bromide CAS:119302-91-9	Rocuronium Bromide is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia to facilitate endotracheal intubation by providing skeletal muscle relaxation.It is used for both standard and rapid sequence induction(RSI).	price>
R-R-4126	CB2R/FAAH modulator-3 CAS No.2876918-67-9	CB2R/FAAH modulator-3 (compound 27)/CAS No.2876918-67-9 is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor. The Ki values for CB2R/FAAH modulator-3 are 20.1 and 67.6 nM for CB2R and CB1R, respectively, and the IC50 value for FAAH is 3.4 μM. CB2R/FAAH modulator-3 can be used in studies related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection.	price>
R-C-2427	Aclidinium Bromide CAS:320345-99-1	Aclidinium bromide is a long-acting anticholinergic bronchodilator approved by the FDA in 2012 for use in the management of chronic obstructive pulmonary disease(COPD)which includes chronic bronchitis and emphysema.	price>
R-R-4127	PGN36 CAS No.1564253-75-3	PGN36 (Compound 18)/CAS No.1564253-75-3 is a selective cannabinoid CB2 receptor (CB2R) antagonist with a Ki of 0.09 µM.	price>
R-C-2428	Otilonium Bromide CAS:26095-59-0	Otilonium bromide is an antimuscarinic and calcium channel blocker used to relieve spasmodic pain of the gut, especially in irritable bowel syndrome.	price>
R-R-4128	AM6545 CAS No.1245626-05-4	AM6545/CAS No.1245626-05-4 is a peripherally active, cannabinoid receptor antagonist with limited brain penetration. AM6545 binds to CB1 and CB2 receptors with Kis of 1.7 nM and 523 nM, respectively. AM6545 is a neutral antagonist. AM6545 can be used for the research of obesity and its complications.	price>
R-C-2429	Gallamine Triethiodide CAS:65-29-2	Gallamine Triethiodide is a mAChR M2 antagonist with pronounced cardioselectivity.It acts by combining with the cholinergic receptor sites in muscle and competitively blocks the transmitter action of acetylcholine.It is a synthetic non-depolarizing blocking drug.	price>
R-R-4129	2-Palmitoylglycerol CAS No.23470-00-0	2-Palmitoylglycerol (2-Palm-Gl)/CAS No.23470-00-0, an congener of 2-arachidonoylglycerol (2-AG), is a modest cannabinoid receptor CB1 agonist. 2-Palmitoylglycerol also may be an endogenous ligand for GPR119.	price>
R-C-2430	Pyridostigmine Bromide CAS:101-26-8	Pyridostigmine Bromide is a cholinesterase inhibitor with a slightly longer duration of action than neostigmine.It is used in the treatment of myasthenia gravis and to reverse the actions of muscle relaxants.Pyridostigmine bromide binds reversibly to acetylcholinesterase active sites in the peripheral nervous system,thereby preventing the breakdown of acetylcholine. This leads to an accumulation of acetylcholine at cholinergic synapses and facilitates transmission of impulses across the neuromuscular junction.	price>
R-R-4130	CB-25 CAS No.869376-63-6	CB-25/CAS No.869376-63-6 is a ligand of CB1 cannabinoid receptors, acting as a partial agonist. CB-25 enhances Forskolin (HY-15371)-induced cAMP formation in cancer cells but not hCB1-CHO cells.	price>
R-C-2431	Rivastigmine Tartrate CAS:129101-54-8	Rivastigmine,also known as ENA-713,is a carbamate-derived reversible cholinesterase inhibitor that is selective for the central nervous system and is used for the treatment of Dementia,Alzheimer is Disease and Parkinson is Disease.It acts by covalently modifying a serine residue in the active site by carbamoylation,as it stabilizes or reduces the rate of decline in certain cognitive functions.	price>
R-R-4131	β-Caryophyllene-d2 CAS No.2006272-96-2	β-Caryophyllene-d2/CAS No.2006272-96-2 is deuterium labeled β-Caryophyllene. β-Caryophyllene is a CB2 receptor agonist.	price>
R-C-2432	Neostigmine Bromide CAS:114-80-7	Neostigmine bromide is a reversible inhibitor of acetylcholinesterase.AChE (acetylcholinesterase)is a hydrolase that hydrolyzes the neurotransmitter acetylcholine at the neuromuscular junction and cholinergic synaspe.It terminates the signal transductions and plays a role in neuronal apoptosis.	price>

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