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Catalog	name	Description	price
R-C-2316	Efonidipine CAS:111011-63-3	Efonidipine(NZ-105)is an L-and T-type calcium channel blocker leading to vasodilation and decreased automaticity of the heart.It also suppresses aldosterone secretion from the adrenal.	price>
R-R-4016	1,2-Bis(4-hexylphenyl)ethane-1,2-dione CAS :869081-44-7	1,2-Bis(4-hexylphenyl)ethane-1,2-dione/CAS :869081-44-7 is an active pharmaceutical ingredient.It finds applic ation in the synthesis of specific dyes, pharmaceutical intermediates(which can be used to prepare MOF ligands), and as a component in the formulation of adhesives or coatings. We can mass produce (kg level), process scaling up, pilot supply, raw material supply, and intermediate production. Our production technology is mature and more cost-effective. Feel free to inquire at any time.	price>
R-C-2317	Panaxadiol CAS:19666-76-3	Panaxadiol(20(R)-Panaxadiol)is a triterpene sapogenin originally found in species of Panax(ginseng)and exhibits anticancer,cardioprotective,anti-arrhythmic,and antioxidative activities.It inhibits Ca2+ channels,decreasing channel open time and open state probability in vitro and displaying anti-arrhythmic potential.	price>
R-R-4017	TRV055 hydrochloride	TRV055 hydrochloride, a G-protein-biased agonist, is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV055 hydrochloride is efficacious in stimulating cellular Gq-mediated signaling.	price>
R-C-2318	CM 4620 CAS:1713240-67-5	CM 4620 is an inhibitor of calcium-release activated calcium-channel(CRAC channel).CM4620 inhibits Orai1/STIM1-mediated Ca2+ currents and Orai2/STIM1-mediated currents with IC50 of near 120 nM and 900 nM.	price>
R-R-4018	TRV056 CAS No.812644-79-4	TRV056/CAS No.812644-79-4 is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV056 is efficacious in stimulating cellular Gq-mediated signaling. TRV056 can be used to develop the Gq-biased AT1R agonists.	price>
R-C-2319	Columbianadin CAS:5058-13-9	Columbianadin(Zosimin,2-Butenoic acid),a natural coumarin from Angelica decursiva,is known to have various biological activities including calcium-channel blocking activity,cytotoxic activity against various cancer cell lines,analgesic activities,intestinal absorption and transportation,anti-inflammatory and anti-cancer effects.	price>
R-R-4019	TRV055 CAS No.25849-90-5	TRV055/CAS No.25849-90-5, a G-protein-biased agonist, is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV055 is efficacious in stimulating cellular Gq-mediated signaling.	price>
R-C-2320	Tetrandrine (NSC-77037) CAS:518-34-3	Tetrandrine(NSC-77037;d-Tetrandrine)is a bis-benzyl-isoquinoline alkaloid,which inhibits voltage-gated Ca2+ current(ICa)and Ca2+-activated K+ current.	price>
R-R-4020	Norleual TFA	Norleual TFA, an angiotensin (Ang) IV analog, is a hepatocyte growth factor (HGF)/c-Met inhibitor with an IC50 of 3 pM. Norleual TFA is an AT4 receptor antagonist and exhibits potent antiangiogenic activities.	price>
R-C-2321	Praeruptorin A CAS:73069-27-9	Praeruptorin A is a main bioactive constituent of Peucedanum praeruptorum(also known as Bai-Hua Qian Hu).Praeruptorin A exerts anti-inflammatory effects in vitro through inhibition of NF-κB activation.	price>
R-R-4021	GSK1820795A CAS No.2650253-86-2	GSK1820795A/CAS No.2650253-86-2, as a telmisartan analog, is a selective hGPR132a antagonist. GSK1820795A blocks activation of yeast cells expressing hGPR132a by N-acylamides. GSK1820795A is also a angiotensin II antagonists and partial PPARγ agonists (compound 38).	price>
R-C-2322	Ginsenoside Rd CAS: 52705-93-8	Ginsenoside Rd(Panaxoside Rd,Sanchinoside Rd),a minor ginseng saponin,has several pharmacological activities such as immunosuppressive activity,anti-inflammatory activity,immunological adjuvant,anti-cancer activity and wound-healing activity.Ginsenoside Rd inhibits TNFα-induced NF-κB transcriptional activity with an IC50 of 12.05±0.82 μM in HepG2 cells.Ginsenoside Rd inhibits expression of COX-2 and iNOS mRNA.Ginsenoside Rd also inhibits Ca2+ influx.	price>
R-R-4022	Azilsartan-d5 CAS No.1346599-45-8	Azilsartan-d5/CAS No.1346599-45-8 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist.	price>
R-C-2323	Rhynchophylline CAS:76-66-4	Rhynchophylline(Mitrinermine),an active component isolated from species of the genus Uncaria,acts as a calcium channel blocker and is widely used in traditional Chinese medicine mainly for treating ailments of central nervous and cardiovascular systems,such as lightheadedness,convulsions,numbness,and hypertension.	price>
R-R-4023	Irbesartan-d4 CAS No.1216883-23-6	Irbesartan-d4/CAS No.1216883-23-6 is the deuterium labeled Irbesartan, which is a highly potent and specific angiotensin II type 1 (AT1) receptor antagonist.	price>
R-C-2324	Levamlodipine CAS:103129-82-4	Levamlodipine((S)-Amlodipine)is a powerful dihydropyridine calcium channel blocker,possessing vasodilation properties and used in the treatment of hypertension and angina.	price>
R-R-4024	Telmisartan-d3 CAS No.1189889-44-8	Telmisartan-d3/CAS No.1189889-44-8 is the deuterium labeled Telmisartan. Telmisartan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM.	price>
R-C-2325	Protopine CAS:130-86-9	Protopine(Corydinine,Fumarine,Biflorine,Macleyine),an alkaloid present in different plants,has been shown to exhibit a number of activities,such as inhibition of calcium influx through both voltage and receptor-operated channels and inhibition of rabbit blood platelet aggregation.It also possesses anti-cholinergic and anti-histaminic as well as anti-bacterial activities.	price>
R-R-4025	Eprosartan mesylate CAS No.144143-96-4	Eprosartan mesylate (SKF-108566J)/CAS No.144143-96-4 is a selective, competitive, nonpeptid and orally active angiotensin II receptor antagonist, used as an antihypertensive. Eprosartan mesylate binds angiotensin II receptor with IC50s of 9.2 nM and 3.9 nM in rat and human adrenal cortical membranes, respectively.	price>

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