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Catalog	name	Description	price
R-R-3898	Brombuterol-d9 CAS No.1353940-55-2	Brombuterol-d9/CAS No.1353940-55-2 is a deuterium labeled Brombuterol. Brombuterol is a β-adrenergic receptor agonist.	price>
R-C-2199	Asciminib (ABL001) CAS:1492952-76-7	Asciminib（ABL001）is a potent allosteric inhibitor of BCR-ABL.ABL001 prevents emergence of resistant disease when administered in combination with nilotinib in an in vivo murine model of chronic myeloid leukemia.Cell proliferation studies demonstrate that ABL001 selectively inhibited the growth of CML and Ph+ ALL cells with potencies ranging from 1-10nM range.	price>
R-C-2289	Apcin CAS:300815-04-7	Apcin(APC inhibitor)is an inhibitor of the E3 ligase activity of the mitotic anaphase-promoting complex/cyclosome(APC/C)that binds to Cdc20 and competitively inhibits the ubiquitylation of D-box-containing substrates.	price>
R-R-3899	Mibenratide CAS No.1239011-83-6	Mibenratide/CAS No.1239011-83-6, a small cyclic peptide, is an adrenergic β1 receptor antagonist. Mibenratide can be used for heart failure research.	price>
R-C-2200	Berbamine CAS:478-61-5	Berbamine(BA),a traditional Chinese medicines extracted from Berberis amurensis (xiaoboan),is a novel inhibitor of bcr/abl fusion gene with potent anti-leukemia activity and also an inhibitor of NF-κB,Berbamine(BA)induces apoptosis in human myeloma cells and inhibits the growth of cancer cells by targeting Ca²⁺/calmodulin-dependent protein kinase II (CaMKII).	price>
R-R-3900	Nadolol-d9 CAS No.94513-92-5	Nadolol-d9/CAS No.94513-92-5 is the deuterium labeled Nadolol. Nadolol is a non-selective and orally active β-adrenergic receptors blocker.	price>
R-C-2201	GMB-475 CAS:2490599-18-1	GMB-475 is a degrader of BCR-ABL1 tyrosine kinase based on PROTAC,overcoming BCR-ABL1-dependent drug resistance.GMB-475 targets BCR-ABL1 protein and recruits the E3 ligase Von Hippel Lindau(VHL),resulting in ubiquitination and subsequent degradation of the oncogenic fusion protein.	price>
R-R-3901	Clorprenaline CAS No.3811-25-4	Clorprenaline/CAS No.3811-25-4 is a potent agonist of β2-adrenergic. Clorprenaline promotes animal muscular mass growth and decreases fat accumulation. Clorprenaline is a potential new lean meat-boosting feed additive.	price>
R-C-2202	Ramucirumab (anti-VEGFR2) CAS:947687-13-0	Ramucirumab is a human VEGFR-2 antagonist for the treatment of solid tumors. Ramucirumab is a recombinant human immunoglobulin G1 monoclonal antibody that binds to the extracellular binding domain of VEGFR-2 and prevents the binding of VEGFR ligands:VEGF-A,VEGF-C,and VEGF-D.	price>
R-R-3902	Salmeterol-d3 CAS No.497063-94-2	Salmeterol-d3/CAS No.497063-94-2 is a deuterium labeled Salmeterol. Salmeterol is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC50s of 9.6, 6.1, and 5.9, respectively.	price>
R-C-2203	Sulfatinib CAS:1308672-74-3	Sulfatinib(HMPL-012)is a potent and highly selective tyrosine kinase inhibitor against VEGFR1/2/3,FGFR1 and CSF1R with IC50s of in a range of 1 to 24nM.	price>
R-R-3903	Guanoxabenz hydrochloride CAS No.23256-40-8	Guanoxabenz (Hydroxyguanabenz) hydrochloride/CAS No.23256-40-8 is an α2 adrenergic receptor agonist, with a Ki of 4000 nM and the fully activated form 40 nM for an α2A adrenoceptor.	price>
R-C-2204	Taxifolin (Dihydroquercetin) CAS:480-18-2	Taxifolin((+)-Dihydroquercetin)exhibits important anti-tyrosinase activity.Taxifolin exhibits significant inhibitory activity against collagenase with an IC50 value of 193.3μM.Taxifolin is an important natural compound with antifibrotic activity.Taxifolin is a free radical scavenger with antioxidant capacity.	price>
R-R-3904	Arbutamine CAS No.128470-16-6	Arbutamine/CAS No.128470-16-6 is a short-acting, potent and nonselective β-adrenoceptor agonist. Arbutamine stimulates cardiac β1-, tracheal β2-, and adiopocyte β3- adrenergic receptors. Arbutamine provides cardiac stress increases heart rate, cardiac contractility, and systolic blood pressure. Arbutamine can be used for cardiac stress agent .	price>
R-C-2205	SU5214 CAS: 186611-04-1	SU5214 is a potent VEGFR2 inhibitor extracted from patent US5834504A,SU5214, has IC50s of 14.8µM(FLK-1)and 36.7µM(EGFR),respectively.	price>
R-R-3905	Efaroxan hydrochloride CAS No.89197-00-2	Efaroxan hydrochloride/CAS No.89197-00-2 is a potent, selective and orally active α2-adrenoceptor antagonist, with antidiabetic activity. Efaroxan hydrochloride is a selective I1-Imidazoline receptor antagonist. Efaroxan hydrochloride can be used for the research of cardiovascular disease.	price>
R-C-2206	SU5408 CAS:15966-93-5	SU5408(VEGFR2 Kinase Inhibitor I)is a potent and cell-permeable inhibitor of VEGFR2 kinase with an IC50 of 70nM.	price>
R-R-3906	NP10679	NP10679 is a selective, pH dependent GluN2B subunit-specific N-methyl-D-aspartate (NMDA) receptor inhibitor with high oral bioavailability and good brain penetration. NP10679 inhibits GluN2B with IC50s of 23 and 142 nM at pH 6.9 and 7.6, respectively. NP10679 is a histamine H1 antagonist and a hERG channel inhibitor with IC50s of 73 and 620 nM, respectively. NP10679 is a reversible inhibitor of human liver CYP enzymes.	price>
R-C-2207	SU5205 CAS:3476-86-6	SU5205 is an inhibitor of VEGFR2 (FLK-1),with an IC50 of 9.6μM.	price>
R-R-3907	Scopine hydrochloride CAS No.85700-55-6	Scopine hydrochloride (6,7-Epoxytropine hydrochloride)/CAS No.85700-55-6 is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.	price>

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