Astemizole CAS: 68844-77-9
Astemizole
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-C-2072 | 100mg | 140.00 | + Add to cart |
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R-C-2072 | 500mg | 400.00 | + Add to cart |
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R-C-2072 | 1g | 700.00 | + Add to cart |
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Product description
Astemizole is a potent antihistamine(H1-receptor antagonist,IC50=4nM)that displays selectivity over dopamine,5-HT,and muscarinic acetylcholine receptors.This compound has shown potent hERG K+ channel blocking activity (IC50=0.9nM),antimalarial activity in multidrug resistant strains in vitro(IC50=227-734nM),and has been used as a chaperone to correct folding defects and restore protein function for some mutated forms of hERG channels.
Appearance | N/A |
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Molecular Weight | N/A |
purity | >95% |
PDI by GPC | <1.5 |
Solubility | N/A |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 3 weeks |
Stability | 1 year |
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