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Catalog	name	Description	price
R-C-1696	NCB-0846 CAS：1792999-26-8	NCB-0846 is the first orally available small-molecule TNIK inhibitor,having anti-Wnt activity and suppressing Wnt-driven intestinal tumorigenesis,also inhibiting FLT3,JAK3,PDGFRa,TRKA,CDK2/CycA2,and HGK.	price>
R-R-3396	Sertindole-d4 CAS No.1794737-42-0	Sertindole-d4/CAS No.1794737-42-0 is the deuterium labeled Sertindole. Sertindole, a neuroleptic, is one of the newer antipsychotic medications available.	price>
R-C-1697	ETP-46321 CAS：1252594-99-2	ETP-46321 is a potent and orally bioavailable PI3Kα and PI3Kδ inhibitor with Kiapps of 2.3 and 14.2 nM,respectively.	price>
R-R-3397	Aripiprazole (1,1,2,2,3,3,4,4-d8) CAS No.1089115-04-7	Aripiprazole (1,1,2,2,3,3,4,4-d8)/CAS No.1089115-04-7 is the deuterium labeled Aripiprazole. Aripiprazole (OPC-14597) is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM.	price>
R-C-1698	Debio 0617B CAS:1332329-27-7	Debio-0617B is a first-in-class multi-kinase inhibitor.Debio-0617B targets pSTAT3,pSTAT5,JAK,SRC,ABL,and class III/V RTKs.	price>
R-R-3398	Paliperidone-d4 CAS No.1020719-55-4	Paliperidone-d4/CAS No.1020719-55-4 is the deuterium labeled Paliperidone. Paliperidone (9-Hydroxyrisperidone), the major active metabolite of Risperidone, is a dopamine D2 antagonist and 5-HT2A antagonist. Paliperidone is also active as an antagonist at α1 and α2 adrenergic receptors and H1-histaminergic receptors. Paliperidone, a antipsychotic agent, shows efficacy against schizophrenia.	price>
R-C-1699	SRT-2104 CAS：1093403-33-8	SRT 2104 is a first-in-class,highly selective and brain-permeable activator of the NAD+dependent deacetylase Sirt1,increases Sirt1 protein,but shows no effect on Sirt1 mRNA.Used in the research of diabetes mellitus and Huntington is disease.	price>
R-R-3399	Alverine-d5 citrate CAS No.1215327-00-6	Alverine-d5 (citrate)/CAS No.1215327-00-6 is the deuterium labeled Alverine citrate.	price>
R-C-1700	Lesinurad CAS： 878672-00-5	Lesinurad is a URAT1 and OAT inhibitor,is determined to be a substrate for the kidney transporters OAT1 and OAT3 with Km values of 0.85 and 2µM, respectively.	price>
R-R-3400	Trazodone-d6 hydrochloride CAS No.1181578-71-1	Trazodone-d6 (hydrochloride)/CAS No.1181578-71-1 is the deuterium labeled Trazodone hydrochloride.	price>
R-C-1701	lusutrombopag CAS：1110766-97-6	Lusutrombopag（S-888711is an orally bioavailable,small molecule thrombopoietin (TPO)receptor agonist being developed by Shionogi for chronic liver disease(CLD) patients with thrombocytopenia prior to elective invasive surgery.	price>
R-R-3401	MS 245 oxalate CAS No.275363-58-1	MS 245 oxalate/CAS No.275363-58-1 is a potent antagonist of 5-HT6 receptor with a Ki of 2 nM.	price>
R-C-1702	Granisetron CAS：109889-09-0	Granisetron(Sancuso,Kevatril,Granisetronum,Sustol)is a serotonin receptor(5HT-3 selective)antagonist that is used as an antiemetic and antinauseant for cancer chemotherapy.	price>
R-R-3402	Blonanserin-d5 CAS No.1346599-86-7	Blonanserin-d5/CAS No.1346599-86-7 is a deuterium labeled Blonanserin. Blonanserin is a dopamine D2/5-HT2 receptor antagonist and an atypical antipsychotic.	price>
R-C-1703	Bestatin CAS: 58970-76-6	Bestatin(NK421,Ubenimex)is a potent aminopeptidase-B and leukotriene(LT)A4 hydrolase inhibitor,used in the treatment of acute myelocytic leukemia.	price>
R-R-3403	SB-216641A CAS No.193611-67-5	SB-216641A (SB-216641 hydrochloride)/CAS No.193611-67-5 is a selective antagonist of 5-HT1B/D receptor. SB-216641A shows high affinity and selectivity for h5-HT1B receptors over h5-HT1D receptors. SB-216641A inhibits the function of SKF-99101H.	price>
R-C-1704	SH5-07 (SH-5-07) CAS:1456632-41-9	SH5-07 is a robust hydroxamic acid-based STAT3 inhibitor,which induce antitumor cell effects in vitro and antitumor response in vivo against human glioma and breast cancer models.	price>
R-R-3404	Cyproheptadine-d3 CAS No.2712455-05-3	Cyproheptadine-d3/CAS No.2712455-05-3 is deuterium labeled Cyproheptadine.	price>
R-C-1705	GNE-3511 CAS:1496581-76-0	GNE-3511 is a potent and selective dual leucine zipper kinase(DLK,MAP3K12) inhibitors with activity in neurodegeneration models.GNE-3511 displays concentration-dependent protection of neurons from degeneration in vitro and demonstrated dose-dependent activity in two different animal models of disease. GNE-3511 displays protection of primary neurons in an in vitro axon degeneration assay as well as activity in the mouse models of glaucoma/optic neuropathy (optic nerve crush)and Parkinson is disease(MPTP)after oral dosing.	price>
R-R-3405	Robalzotan hydrochloride CAS No.184674-99-5	Robalzotan hydrochloride (NAD-299 hydrochloride)/CAS No.184674-99-5 is a potent and selective 5-Hydroxytryptamine 1A (5-HT1A) inhibitor. Robalzotan hydrochloride increases the firing rate of 5-HT cells. Robalzotan hydrochloride induces 5-HT1A receptor occupancy. Robalzotan hydrochloride has the potential for the research of a cholinergic deficit in the central -nervous system.	price>

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