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Catalog	name	Description	price
R-C-1455	Betahistine CAS:5638-76-6	Betahistine is a histamine analog and H1 receptor agonist that serves as a vasodilator.It is used in MENIERE DISEASE and in vascular headaches but may exacerbate bronchial asthma and peptic ulcers.Betahistine dihydrochloride is an anti-vertigo drug.It is commonly prescribed for balance disorders or to alleviate vertigo symptoms associated with Ménière is disease.It was first registered in Europe in 1970 for the treatment of Ménière is disease.	price>
R-R-3155	Setiptiline maleate CAS No.85650-57-3	Setiptiline maleate (MO-8282 maleate)/CAS No.85650-57-3 is a serotonin receptor antagonist. Setiptiline maleate is a tetracyclic antidepressant (TeCA) which acts as a noradrenergic and specific serotonergic antidepressant (NaSSA). Setiptiline maleate acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, likely at the 5-HT2A, 5-HT2C, and/or 5-HT3 subtypes, as well as an H1 receptor inverse agonist/antihistamine.	price>
R-C-1456	NSC19005(Betahistine EP Impurity C) CAS:5452-87-9	Betahistine EP Impurity C(NSC19005)is an impurity of Betahistine.Betahistine is a potent,orally active and well-tolerated histamine H1 receptor agonist and H3 receptor antagonist used for the study of rheumatoid arthritis(RA).	price>
R-R-3156	Lumateperone tosylate CAS No.1187020-80-9	Lumateperone (ITI-007) tosylate/CAS No.1187020-80-9 is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a dopamine D1 receptor modulator. Lumateperone tosylate has anticancer activity and can also be used in studies of psychiatric disorders such as schizophrenia.	price>
R-C-1457	NKL 22 CAS:537034-15-4	NKL 22 is a HDAC inhibitor.The value of IC 50 is 78 uM NKL 22 increase frataxin protein concentrations NKL 22 inhibitors increase FXN mRNA in FRDA lymphocytes. HDAC inhibitors act directly on FXN.	price>
R-R-3157	(Z)-Thiothixene CAS No.3313-26-6	(Z)-Thiothixene/CAS No.3313-26-6 is an antagonist of serotonergic receptor extracted from patent US 20150141345 A1.	price>
R-C-1458	FPS-ZM1 CAS:945714-67-0	FPS-ZM1 is a blood-brain-barrier permeant,non-toxic,tertiary amide compound which is a high affinity RAGE-specific inhibitor,blocking Aβ binding to the V domain of RAGE.	price>
R-R-3158	Eletriptan hydrobromide CAS No.177834-92-3	Eletriptan hydrobromide (Eletriptan HBr)/CAS No.177834-92-3 is a selective 5-HT1B and 5-HT1D receptor agonist with Ki of 0.92 nM and 3.14 nM, respectively.	price>
R-C-1459	PYRACLONIL CAS：158353-15-2	Pyraclonil is a proporphyrinogen oxidase(PPO)inhibitor.Pyraclonil is a herbicide agent and is highly effective in controlling the susceptible(S)and multiple-herbicide-resistant(MHR)E.indica populations.	price>
R-R-3159	SB 258719 CAS No.195199-95-2	SB 258719/CAS No.195199-95-2 is a selective 5-HT7 receptor antagonist with high affinity (pKi=7.5) for the receptor. SB 258719 can be used for the research of cancer and neurological disease.	price>
R-C-1460	Mitoquinone CAS:444890-41-9	Mitoquinone is a mitochondria-targeted antioxidant designed to accumulate within mitochondria in vivo in order to protect against oxidative damage.	price>
R-R-3160	Ziprasidone hydrochloride monohydrate CAS No.138982-67-9	Ziprasidone (CP-88059) hydrochloride monohydrate/CAS No.138982-67-9 is an orally active combined 5-HT and dopamine receptor antagonist. Ziprasidone hydrochloride monohydrate has affinities for Rat D2 (Ki=4.8 nM), 5-HT2A (Ki=0.42 nM) and 5-HT1A (Ki=3.4 nM).	price>
R-C-1461	ASC-J9 CAS:52328-98-0	Dimethylcurcumin(ASC-J9,Dimethyl curcumin,GO-Y025)is an androgen receptor (AR)degradation enhancer that suppresses castration-resistant prostate cancer growth through degradation of full-length and splice variant androgen receptors.	price>
R-R-3161	Jatrorrhizine hydroxide CAS No.483-43-2	Jatrorrhizine hydroxide/CAS No.483-43-2 is an alkaloid isolated from Coptis chinensis with neuroprotective, antimicrobial, antiplasmodial and antioxidant activities. Jatrorrhizine hydroxide is a potent and orally active inhibitor of AChE (IC50=872 nM) over >115-fold selectivity for BuChE. Jatrorrhizine hydroxide reduces uptake of serotonin (5-HT) and norepinephrine (NE) via inhibition of uptake-2 transporters.	price>
R-C-1462	PCI 34051 CAS:950762-95-5	PCI-34051 is a potent and specific HDAC8 inhibitor with IC50 of 10 nM in a cell-free assay.It has greater than 200-fold selectivity over HDAC1 and 6, more than 1000-fold selectivity over HDAC2,3,and 10.PCI-34051 induces caspase-dependent apoptosis.	price>
R-R-3162	Gepirone CAS No.83928-76-1	Gepirone/CAS No.83928-76-1 is a selective and affinitive 5-HT1A agonist. Gepirone binds selectively to 5-HT1A receptor binding site. Gepirone acts as an antidepressant agent can be used for anxiety and major depressive disorder research.	price>
R-C-1463	Bohemine CAS:189232-42-6	Bohemine is a potent and selective,cell-permeable,cyclin-dependent kinase(CDK) inhibitor with IC50=1 µM.Bohemine is structurally similar to Olomoucine and Roscovitine.	price>
R-R-3163	Asenapine CAS No.65576-45-6	Asenapine (Org 5222)/CAS No.65576-45-6, an atypical antipsychotic, is an antagonist of serotonin receptors (pKi: 8.4-10.5), adrenoceptors (pKi: 8.9-9.5), dopamine receptors (pKi: 8.9-9.4) and histamine receptors (pKi: 8.2-9.0). Asenapine can be used in the research of schizophrenia and bipolar disorder.	price>
R-C-1464	TA 01 CAS:1784751-18-3	TA-01 is an inducer of cardiomyocyte differentiation from human embryonic stem cells following mesoderm induction.	price>
R-R-3164	RU 24969 CAS No.66611-26-5	RU 24969/CAS No.66611-26-5 is a preferential 5-HT1B agonist, with a Ki of 0.38 nM, but also displays appreciable affinity for the 5-HT1A receptor (Ki=2.5 nM), and has low affinity for other receptor sites in the brain. RU 24969 could decrease fluid consumption and increase forward locomotion.	price>

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