Vercirnon sodium CAS No.886214-18-2
Vercirnon sodium CAS No.886214-18-2
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-4206 | 5mg | 490.00 | + Add to cart |
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R-R-4206 | 10mg | 730.00 | + Add to cart |
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Product description
Vercirnon (GSK1605786A) sodium/CAS No.886214-18-2 is an orally bioavailable, selective, and potent antagonist of CCR9. Vercirnon sodium inhibits CCR9-mediated Ca2+ mobilization and chemotaxis on Molt-4 cells with IC50 values of 5.4 and 3.4 nM, respectively. Vercirnon sodium is selective for CCR9 over CCR1-12 and CX3CR1-7 (IC50s>10 µM for all). Vercirnon sodium is an equipotent inhibitor of CCL25-directed chemotaxis of both splice forms of CCR9 (CCR9A and CCR9B) with IC50 values of 2.8 and 2.6 nM, respectively.
Appearance | N/A |
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Molecular Weight | 466.91 |
Purity | >90% |
CAS | 886214-18-2 |
Formula | C22H20ClN2NaO4S |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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