SB-277011 hydrochloride CAS No.215804-67-4
SB-277011 hydrochloride CAS No.215804-67-4
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-3186 | 25mg | 280.00 | + Add to cart |
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R-R-3186 | 50mg | 460.00 | + Add to cart |
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Product description
SB-277011 hydrochloride (SB-277011A hydrochloride)/CAS No.215804-67-4 is a potent, selective, orally bioavailable and brain penetrate dopamine D3 receptor (D3R) antagonist with Ki values of 10.7 nM and 11.2 nM at rodent and human D3R, respectively. SB-277011 hydrochloride displays 80- to 100-fold selectivity over other dopamine receptors with pKis of 8.0, 6.0, <5.2, and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively.
Appearance | N/A |
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Molecular Weight | 475.02 |
Purity | >90% |
CAS | 215804-67-4 |
Formula | C28H31ClN4O |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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