S1RA hydrochloride CAS No.1265917-14-3
S1RA hydrochloride CAS No.1265917-14-3
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-3118 | 25mg | 330.00 | + Add to cart |
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R-R-3118 | 50mg | 540.00 | + Add to cart |
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Product description
S1RA (E-52862) hydrochloride/CAS No.1265917-14-3 is an orally active and selective sigma-1 receptor (σ1R) antagonist with a Ki value of 17 nM. S1RA hydrochloride shows good selectivity against σ2R (Ki >1000 nM). S1RA hydrochloride is a human 5-HT2B receptor antagonist with an IC50 value of 4.7 μM. S1RA hydrochloride inhibits neuropathic pain and activity-induced spinal sensitization.
Appearance | N/A |
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Molecular Weight | 373.88 |
Purity | >90% |
CAS | 1265917-14-3 |
Formula | C20H24ClN3O2 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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