Home > products > fluorescent-dyes
> No-ROS-Rox-derivatives
> par2-1-6-amide-human-trifluoroacetate-salt
PAR2 (1-6) amide (human) (trifluoroacetate salt),cas:2379569-17-0
(S)-6-amino-2-(2-((2S,3S)-2-((S)-2-((S)-2-amino-3-hydroxypropanamido)-4-methylpentanamido)-3-methylpentanamido)acetamido)-N-((S)-1-amino-3-methyl-1-oxobutan-2-yl)hexanamide, trifluoroacetate salt
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
---|---|---|---|---|
R-XASYS-00122 | 25mg | 460.00 | + Add to cart |
|
R-XASYS-00122 | 50mg | 875.00 | + Add to cart |
|
|
Product description
PAR2 (1-6) amide(C28H54N8O7·XCF3COOH,614.8) is a synthetic peptide agonist of proteinase-activated receptor 2 (PAR2) that corresponds to residues 1-6 of the amino terminal tethered ligand sequence of human PAR2 and residues 37-42 of the full-length sequence.It binds to NCTC 2544 cells expressing human PAR2 (Ki = 9.64 µM in a radioligand binding assay) and induces calcium mobilization in the same cells (EC50 = 0.075 µM).PAR2 (1-6) amide (100 µM) reduces colony formation of A549 lung cancer cells.
Appearance | N/A |
---|---|
Molecular Weight | N/A |
Purity | >90% |
Solubility | N/A |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 3 weeks |
Stability | 1 year |
Document
Related Product