NAS-181 dimesylate CAS No.1217474-40-2
NAS-181 dimesylate CAS No.1217474-40-2
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-3146 | 10mg | 290.00 | + Add to cart |
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R-R-3146 | 25mg | 600.00 | + Add to cart |
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Product description
NAS-181 dimesylate/NAS181/CAS No.1217474-40-2 is a potent and selective antagonist of rat 5-HT1B receptor, with a Ki of 47 nM. NAS181 shows 13-fold selectivity for r5-HT1B over bovine 5-HT1B receptor (Ki=630 nM). NAS181 increases the 5-HT turnover and the synaptic concentration of 5-HT by inhibiting terminal r5-HT1B autoreceptors.
Appearance | N/A |
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Molecular Weight | 538.63 |
Purity | >90% |
CAS | 1217474-40-2 |
Formula | C21H34N2O10S2 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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