Inobrodib CAS No.2222941-37-7
Inobrodib CAS No.2222941-37-7
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-2429 | 10mg | 330.00 | + Add to cart |
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R-R-2429 | 25mg | 670.00 | + Add to cart |
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Product description
Inobrodib (CCS1477)/CAS No.2222941-37-7 is an orally active, potent, and selective inhibitor of the p300/CBP bromodomain. Inobrodib binds to p300 and CBP with Kd values of 1.3 and 1.7 nM, respectively, and with 170/130-fold selectivity compared with BRD4 with a Kd of 222 nM. CCS1477 inhibits cell proliferation in prostate cancer cell lines and decreases androgen receptor (AR)- and C-MYC-regulated gene expression.
Appearance | N/A |
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Molecular Weight | 534.60 |
Purity | >90% |
CAS | 2222941-37-7 |
Formula | C30H32F2N4O3 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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