GSK8814 CAS No.1997369-78-4
GSK8814 CAS No.1997369-78-4
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-2520 | 5mg | 430.00 | + Add to cart |
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R-R-2520 | 10mg | 760.00 | + Add to cart |
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Product description
GSK8814/CAS No.1997369-78-4 is a potent, selective, and ATAD2/2B bromodomain chemical probe and inhibitor, with a binding constant pKd=8.1 and a pKi=8.9 in BROMOscan. GSK8814 binds to ATAD2 and BRD4 BD1 with pIC50s of 7.3 and 4.6, respectively. GSK8814 shows 500-fold selectivity for ATAD2 over BRD4 BD1.
Appearance | N/A |
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Molecular Weight | 527.61 |
Purity | >90% |
CAS | 1997369-78-4 |
Formula | C28H35F2N5O3 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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