GNE-207 CAS No.2158266-58-9
GNE-207 CAS No.2158266-58-9
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
---|---|---|---|---|
R-R-2510 | 5mg | 320.00 | + Add to cart |
|
R-R-2510 | 10mg | 530.00 | + Add to cart |
|
|
Product description
GNE-207/CAS No.2158266-58-9 is a potent, selective and orally bioavailable inhibitor of the bromodomain of CBP, with an IC50 of 1 nM, exhibits a selectively index of >2500-fold against BRD4 (1). GNE-207 shows excellent CBP potency, with an EC50 of 18 nM for MYC expression in MV-4-11 cells.
Appearance | N/A |
---|---|
Molecular Weight | 510.59 |
Purity | >90% |
CAS | 2158266-58-9 |
Formula | C29H30N6O3 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
Document
Related Product