GNE-064 CAS No.1997321-20-6
GNE-064 CAS No.1997321-20-6
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-2502 | 5mg | 280.00 | + Add to cart |
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R-R-2502 | 10mg | 460.00 | + Add to cart |
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Product description
GNE-064 (compound 5)/CAS No.1997321-20-6 is a selective, orally active and highly soluble inhibitor of SMARCA4, SMARCA2 and PBRM1 bromodomains 5. GNE-064 inhibits SMARCA4 with an IC50 of 0.035 μM and inhibits SMARCA2 with an EC50 of 0.10 μM. GNE-064 possess Kds with 0.01, 0.016, 0.018 and 0.049 μM for SMARCA4, SMARCA2, PBRM1 bromodomains 5 and PBRM1 bromodomains 2, repectively. GNE-064 can be used as a chemical probe for the research of agent synthesis.
Appearance | N/A |
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Molecular Weight | 327.38 |
Purity | >90% |
CAS | 1997321-20-6 |
Formula | C17H21N5O2 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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