CXCR2-IN-2 CAS No.1838123-21-9
CXCR2-IN-2 CAS No.1838123-21-9
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-4268 | 5mg | 570.00 | + Add to cart |
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R-R-4268 | 10mg | 1000.00 | + Add to cart |
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Product description
CXCR2-IN-2/CAS No.1838123-21-9 is a selective, brain penetrant, and orally bioavailable CXCR2 antagonist (IC50=5.2 nM/1 nM in β-arrestin assay/CXCR2 Tango assay, respectively). CXCR2-IN-2 displays ~730-fold selectivity over CXCR1 and >1900-fold selectivity over all other chemokine receptors. CXCR2-IN-2 inhibits human whole blood Gro-α induced CD11b expression with an IC50 of 0.04 μM.
Appearance | N/A |
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Molecular Weight | 414.90 |
Purity | >90% |
CAS | 1838123-21-9 |
Formula | C18H23ClN2O5S |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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