CH5138303 cas:959763-06-5
CH5138303
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-C-1010 | 2mg | 100.00 | + Add to cart |
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R-C-1010 | 5mg | 180.00 | + Add to cart |
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R-C-1010 | 10mg | 325.00 | + Add to cart |
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Product description
CH5138303 is a triazine Hsp90 inhibitor.1 CH5138303 binds to the N-terminus of Hsp90α(Kd= 0.52 nM)and inhibits growth of HCT116 and NCI-N87 human tumor cell lines in vitro(IC50s=89 and 66 nM,respectively).CH5138303 also inhibits growth of human NCI-N87 gastric cancer xenografts(ED50=3.9 mg/kg) and displays high oral bioavailability in mice.
Appearance | N/A |
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Molecular Weight | N/A |
purity | >95% |
PDI by GPC | <1.5 |
Solubility | N/A |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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