CF53 CAS No.1808160-52-2
CF53 CAS No.1808160-52-2
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-2580 | 5mg | 430.00 | + Add to cart |
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R-R-2580 | 10mg | 740.00 | + Add to cart |
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Product description
CF53/CAS No.1808160-52-2 is a highly potent, selective and orally active inhibitor of BET protein, with a Ki of <1 nM, Kd of 2.2 nM and an IC50 of 2 nM for BRD4 BD1. CF53 binds to both the BD1 and BD2 domains of BRD2, BRD3, BRD4, and BRDT BET proteins with high affinities, very selective over non-BET bromodomain-containing proteins. CF53 shows potent anti-tumor activity both in vitro and in vivo.
Appearance | N/A |
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Molecular Weight | 443.50 |
Purity | >90% |
CAS | 1808160-52-2 |
Formula | C24H25N7O2 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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