CCG258208 hydrochloride
CCG258208 hydrochloride
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-2924 | 5mg | 330.00 | + Add to cart |
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R-R-2924 | 10mg | 540.00 | + Add to cart |
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Product description
CCG258208 (GRK2-IN-1) hydrochloride is a potent and selective GRK2 (G protein-coupled receptor kinase 2) inhibitor (IC50=30 nM) while maintaining 230-fold selectivity over GRK5 (IC50=7.09 μM) and more than 2500-fold selectivity over GRK1 (IC50=87.3 μM), PKA, and ROCK1. CCG258208 hydrochloride can be used in heart failure research.
Appearance | N/A |
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Molecular Weight | 488.94 |
Purity | >90% |
Synonyms | GRK2-IN-1 hydrochloride |
Formula | C24H26ClFN4O4 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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