AVN-492,cas:1220646-23-0
3-(benzenesulfonyl)-2-N,6-N,6-N,5,7-pentamethylpyrazolo[1,5-a]pyrimidine-2,6-diamine
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-XASYS-00730 | 1mg | 322.00 | + Add to cart |
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R-XASYS-00730 | 5mg | 868.00 | + Add to cart |
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Product description
AVN-492(C17H21N5O2S,359.4) is an antagonist of the serotonin (5-HT) receptor subtype 5-HT6 (Ki = 0.09 nM). It selectively inhibits the 5-HT6 receptor over the 5-HT2B receptor (IC50s = 0.19 and 268 nM, respectively, in a radioligand binding assay). AVN-492 inhibits increases in cAMP levels induced by 5-HT in HEK293 cells expressing the 5-HT6 receptor (IC50 = 1.5 nM).
Appearance | N/A |
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Molecular Weight | N/A |
Purity | >90% |
Solubility | N/A |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 3 weeks |
Stability | 1 year |
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