ABT-639 CAS:1235560-28-7
ABT-639
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-C-1526 | 100mg | 825.00 | + Add to cart |
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R-C-1526 | 200mg | 1200.00 | + Add to cart |
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R-C-1526 | 500mg | 2385.00 | + Add to cart |
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Product description
ABT-639 is a potent and selective T-type calcium channel blocker.ABT-639 effectively reduces nociceptive and neuropathic pain in rats.ABT-639 produces robust antinociceptive activity in experimental pain models at doses that do not significantly alter psychomotor or hemodynamic function in the rat.ABT-639 was significantly less active at other Ca²⁺channels(e.g.Ca(v)1.2 and Ca(v)2.2) (IC50>30μM).ABT-639 has high oral bioavailability(%F=73),low protein binding(88.9%)and a low brain:plasma ratio(0.05:1)in rodents.
Appearance | N/A |
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Molecular Weight | N/A |
purity | >95% |
PDI by GPC | <1.5 |
Solubility | N/A |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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