Product peptide-Inhibitory-peptide

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Catalog	name	Description	price
R-R-0911	D-Pro-Phe-Arg-Chloromethylketone	D-Pro-Phe-Arg-Chloromethylketone/CAS No.88546-74-1, a inhibitor of coagulation factor XII and plasma kallikrein, plays an important role in thrombosis and inflammation.	price>
R-R-0912	GLP-1(32-36)amide	GLP-1(32-36)amide/CAS No.1417302-71-6, a pentapeptide, derived from the C terminus of the glucoregulatory hormone GLP-1. GLP-1(32-36)amide could inhibit weight gain and modulate whole body glucose metabolism in diabetic mice.	price>
R-R-0915	Hemorphin-7	Hemorphin-7/Cas.152685-85-3 is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin. Hemorphin peptides exhibits antinociceptive and antihypertensive activities, activating opioid receptors and inhibiting angiotensin-converting enzyme (ACE).	price>
R-R-0918	Obtustatin triacetate	Obtustatin triacetate is a 41-residue non-RGD disintegrin. Obtustatin triacetate can be isolated from the venom of Vipera lebetina obtusa. Obtustatin triacetate is a potent and selective inhibitor of integrin α1β1 adhesion to type IV collagen. Obtustatin triacetate inhibits angiogenesis and may be used in cancer research.	price>
R-R-0919	Disitertide diammonium	Disitertide (P144) diammonium is a peptidic transforming growth factor-beta 1 (TGF-β1) inhibitor specifically designed to block the interaction with its receptor. Disitertide diammonium is also a PI3K inhibitor and an apoptosis inducer.	price>
R-R-0921	Dihydrocyclosporin A	Dihydrocyclosporin A/CAS.59865-15-5 is a derivative of Cyclosporine A (HY-B0579). Dihydrocyclosporin A significantly inhibites promastigotes and intracellular amastigotes. Dihydrocyclosporin A is highly cytotoxic.	price>
R-R-0925	w-Conotoxin MVIIC TFA	ω-Conotoxin MVIIC TFA is a N- and P/Q-type Ca2+ channel blocker, significantly suppresses the 11-keto-βboswellic acid-mediated inhibition of glutamate release.	price>
R-R-0926	BQ-3020 ammonium	BQ-3020 ammonium is a selective endothelin receptor (ETB receptor) agonist. BQ-3020 ammonium inhibits [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM. BQ-3020 ammonium elicits vasoconstriction in the rabbit pulmonary artery. BQ-3020 ammonium makes relaxation of the pig urinary bladder neck and can be used for cardiovascular disease research.	price>
R-R-0930	GLP-1(28-36)amide	GLP-1(28-36)amide/CAS.1225021-13-5, a C-terminal nonapeptide of GLP-1, is a major product derived from the cleavage of GLP-1 by the neutral endopeptidase (NEP). GLP-1(28-36)amide is an antioxidant and targets to mitochondrion, inhibits mitochondrial permeability transition (MPT). GLP-1(28-36)amide has anti-diabetic and cardioprotection effects.	price>
R-R-0934	Lys-[Des-Arg9]Bradykinin TFA	Lys-[Des-Arg9]Bradykinin TFA/CAS.2763588-90-3, a naturally occurring kinin, is a potent and highly selective bradykinin B1 receptor agonist with a Ki of 0.12 nM, 1.7 nM and 0.23 nM for human, mouse and rabbit B1 receptors, respectively. Lys-[Des-Arg9]Bradykinin TFA has low inhibitory activity on B2 receptors.	price>

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