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Catalog | name | Description | price |
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R-R-4750 | SCR7 CAS No.1533426-72-0 | SCR7/CAS No.1533426-72-0 is an unstable form that can be autocyclized into a stable form SCR7 pyrazine. SCR7 pyrazine is a DNA ligase IV inhibitor that blocks nonhomologous end-joining (NHEJ) in a ligase IV-dependent manner. SCR7 pyrazine is also a CRISPR/Cas9 enhancer which increases the efficiency of Cas9-mediated homology-directed repair (HDR). SCR7 pyrazine induces cell apoptosis and has anticancer activity. | price> |
R-C-3081 | JI-101 CAS NO. 900573-88-8 | JI-101 is an orally active inhibitor of vascular endothelial growth factor receptor 2 (VEGFR2), platelet-derived growth factor receptor beta (PDGFRβ), and the ephrin B4 receptor B4 (EphB4) with potential antiangiogenic and antineoplastic activities.Only for scientific research, not for human body. | price> |
R-R-4751 | Deoxycytidine triphosphate CAS No.2056-98-6 | Deoxycytidine triphosphate (dCTP)/CAS No.2056-98-6 is a nucleoside triphosphate that can be used for DNA synthesis. Deoxycytidine triphosphate has many applications, such as real-time PCR, cDNA synthesis, and DNA sequencing. | price> |
R-C-3082 | SU1498 CAS:168835-82-3 | SU1498, a powerful inhibitor of KDR (IC50=0.7μM), stimulates accumulation of phosphorylated ERK1/2 in endothelial cells.Only for scientific research, not for human body. | price> |
R-R-4752 | Novobiocin CAS No.303-81-1 | Novobiocin (Albamycin)/CAS No.303-81-1 is a potent and orally active antibiotic. Novobiocin also is a DNA gyrase inhibitor and a heat shock protein 90 (Hsp90) antagonist. Novobiocin has the potential for the research of highly beta-lactam-resistant pneumococcal infections. Novobiocin shows anti-orthopoxvirus activity.The free form of the compound is prone to instability, it is advisable to consider the stable salt form (Novobiocin sodium) that retains the same biological activity. | price> |
R-C-3083 | GW806742X CAS:579515-63-2 | GW806742X is a Mixed Lineage Kinase Domain-Like protein (MLKL)inhibitor which binds the MLKL pseudokinase domain with a Kd value of 9.3μM and has anti-necroptosis activity.GW806742X has activity against VEGFR2. Only for scientific research, not for human body. | price> |
R-R-4753 | Crisnatol CAS No.96389-68-3 | Crisnatol (BWA770U)/CAS No.96389-68-3 is an orally active and anticancer agent, and a member of the arylmethylaminopropanediol class of DNA intercalators. Crisnatol shows in vitro cytotoxicity against human breast cancer cells, but not normal human skin fibroblasts. | price> |
R-C-3084 | GW842166X CAS:666260-75-9 | GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM,shows no significant activity at CB1 receptor.Only for scientific research, not for human body. | price> |
R-R-4754 | Herboxidiene CAS No.142861-00-5 | Herboxidiene (GEX1A)/CAS No.142861-00-5 is a potent phytotoxic polyketide from Streptomyces sp. A7847 with a diverse range of activities, including herbicidal, anti-cholesterol, anti-tumor effects. Herboxidiene inhibits the pre-mRNA splicing process by binding to spliceosome-associated protein (SAP) 155, a subunit of SF3b, in the splicesome. | price> |
R-C-3085 | EG00229 CAS:1018927-63-3 | EG00229 is a Neuropilin 1(NRP1)receptor antagonist. EG00229 inhibits VEGFA binding to NRP1.Only for scientific research, not for human body. | price> |
R-R-4755 | 5-PA-dUTP CAS No.179101-49-6 | 5-PA-dUTP (5-Propargylamino-dUTP)/CAS No.179101-49-6 is a C5-modified nucleotide and can be incorporated into DNA nanoparticles (DNPs) for photosensitizer delivery. 5-PA-dUTP is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups. | price> |
R-C-3086 | R1530 CAS:882531-87-5 | R1530 is a pyrazolobenzodiazepine small molecule with potential antiangiogenesis and antineoplastic activities.Only for scientific research, not for human body. | price> |
R-R-4756 | NSC 80467 CAS No.101982-51-8 | NSC 80467/CAS No.101982-51-8, a DNA damaging agent, selectively inhibits survivin. NSC 80467 preferentially inhibits DNA synthesis and results in induction of γH2AX and pKAP1, two markers of DNA damage. | price> |
R-C-3087 | SUN11602 CAS:704869-38-5 | SUN11602 is a small synthetic compound that mimics the neuroprotective activities of bFGF and activates key molecules in the FGF receptor-1-mitogen-activated protein kinase/extracellular signal-regulated kinase-1/2 kinase (FGFR-1-MEK/ERK) signaling pathway.Only for scientific research, not for human body. | price> |
R-R-4757 | MC-VC-PAB-Cyclohexanediamine-Thailanstatin A CAS No.1609108-96-4 | MC-VC-PAB-Cyclohexanediamine-Thailanstatin A/CAS No.1609108-96-4 is a Spliceostatin (HY-16466) analog, and a drug-linker conjugates for ADC, consisting of ADC Cytotoxin Thailanstatin A (HY-129589) and cleavable ADC linker (MC-vc-PAB). MC-VC-PAB-Cyclohexanediamine-Thailanstatin A can be used for ADC synthesis. | price> |
R-C-3088 | SU4312 CAS: 5812-07-7 | SU-4312, also known as DMBI, is a potent and selective inhibitor of VEGFR and PDGFR tyrosine kinases (IC50 values are 0.8 and 19.4 μM respectively).Only for scientific research, not for human body. | price> |
R-R-4758 | FAICAR CAS No.13018-54-7 | FAICAR (5-Formamidoimidazole-4-carboxamide ribotide)/CAS No.13018-54-7 is a purine nucleotide. | price> |
R-C-3089 | CEP-11981 cas: 856691-93-5 | CEP-11981(ESK981)is an orally bioavailable inhibitor of vascular endothelial growth factor receptor (VEGFR) and Tie2 receptor tyrosine kinases with potential antiangiogenic and antineoplastic activities. Only for scientific research, not for human body. | price> |
R-R-4759 | Cytarabine-d2 CAS No.40632-26-6 | Cytarabine-d2/CAS No.40632-26-6 is the deuterium labeled Cytarabine. Cytarabine, a nucleoside analog, causes S phase cell cycle arrest and inhibits DNA polymerase. Cytarabine inhibits DNA synthesis with an IC50 of 16 nM. Cytarabine has antiviral effects against HSV. | price> |
R-C-3090 | Tyrphostin 9 CAS:10537-47-0 | Tyrphostin 9 (SF 6847, RG-50872) is firstly designed as an EGFR inhibitor with IC50 of 460 μM, but is also found to be more potent to PDGFR with IC50 of 0.5 μM.Only for scientific research, not for human body. | price> |