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Catalog	name	Description	price
R-R-4494	LH846 CAS No.639052-78-1	LH846/CAS No.639052-78-1 is a selective inhibitor of CKIδ, with an IC50 of 290 nM, and less potently inhibits CKIα and CKIε, with IC50s of 2.5 μM and 1.3 μM, respectively.	price>
R-C-2795	Alcaftadine (R89674) CAS:147084-10-4	Alcaftadine(R89674)is a histamine H1 receptor antagonist,which is used to prevent eye irritation brought on by allergic conjunctivitis.Alcaftadine is a broad-spectrum antihistamine displaying a high affinity for histamine H1 and H2 receptors and a lower affinity for H4 receptors.Alcaftadine also exhibits modulatory action on immune cell recruitment and mast cell stabilizing effects.	price>
R-C-3325	DSPE-PEG550-BTC	In order to improve the accumulation of anticancer drugs in tumor and enhance the possibility of intracellular delivery,the stealth liposomes modified with arginine glycine aspartic acid (RGD) mimics were used as targeting vectors. Integrin was synthesized and covalently coupled with active polyethylene glycol phospholipid(DSPE-PEG-BTC) to form rgdm coupling compound (DSPE-PEG-RGDM).The binding of melanoma cells to dspe-peg-rgdm was studied by pH sensitive probe bcecf-am.	price>
R-R-4495	Casein Kinase II Inhibitor IV CAS No.863598-09-8	Casein Kinase II Inhibitor IV/CAS No.863598-09-8 is a potent, ATP-competitive of casein kinase II inhibitor with an IC50 of 9 nM. Casein Kinase II Inhibitor IV ia also a human keratinocytes (NHEK) differentiation inducer.	price>
R-C-2796	Maropitant CAS:147116-67-4	Maropitant is a neurokinin(NK1)receptor antagonist.IC50 value:Target:NK1 receptor Maropitant is the first NK1 receptor antagonist developed to treat and prevent emesis in dogs.	price>
R-C-3326	DSPE-PEG750-BTC	In order to improve the accumulation of anticancer drugs in tumor and enhance the possibility of intracellular delivery,the stealth liposomes modified with arginine glycine aspartic acid (RGD) mimics were used as targeting vectors. Integrin was synthesized and covalently coupled with active polyethylene glycol phospholipid(DSPE-PEG-BTC) to form rgdm coupling compound (DSPE-PEG-RGDM).The binding of melanoma cells to dspe-peg-rgdm was studied by pH sensitive probe bcecf-am.	price>
R-R-4496	MU1742	MU1742 is a probe for CK1δ and CK1ε protein kinases.	price>
R-C-2797	L-732,138 CAS:148451-96-1	L-732138 is a selective,potent and competitive neurokinin-1(NK-1)receptor antagonist with an IC50 of 2.3nM.L-732138 has 200-fold more potent in cloned human NK-1 receptors than cloned rat NK-1 receptors,and has>1000-fold more potent than human NK-2 and NK-3 receptors.L-732138 can reduce hyperalgesia and has antitumor action.	price>
R-C-3327	DSPE-PEG350-psCPP	(DSPE) polyethyleneglycol is a combination of phospholipid and polyethylene glycol,which has hydrophilicity and hydrophobicity.Polyethylene glycol liposomes were used to form high-quality materials.It can be used for drug delivery,gene transfection and vaccine delivery.Pegylated phospholipids can significantly improve blood circulation time and stabilize drug encapsulation.These materials can also be used for targeted drug delivery by modifying the ligand with the target surface to add antibodies and peptides.	price>
R-R-4497	PI-828 CAS No.942289-87-4	PI-828/CAS No.942289-87-4 is a dual PI3K and casein kinase 2 (CK2) inhibitor with IC50s of 173 nM, 149 nM, and 1127 nM for p110α, CK2, and CK2α2 in lipid kinase assay, respectively.	price>
R-C-2798	Pizotifen CAS:15574-96-6	Pizotifen is a serotonin antagonist which acts mainly at the 5-HT1,5-HT2A,and 5HT2C receptors with some antihistamine activity.	price>
R-C-3328	DSPE-PEG550-psCPP	(DSPE) polyethyleneglycol is a combination of phospholipid and polyethylene glycol,which has hydrophilicity and hydrophobicity.Polyethylene glycol liposomes were used to form high-quality materials.It can be used for drug delivery,gene transfection and vaccine delivery.Pegylated phospholipids can significantly improve blood circulation time and stabilize drug encapsulation.These materials can also be used for targeted drug delivery by modifying the ligand with the target surface to add antibodies and peptides.	price>
R-R-4498	Casein Kinase 2 Substrate Peptide CAS No.132176-35-3	Casein Kinase 2 Substrate Peptide is a common CK2 substrate peptide. Casein Kinase 2 Substrate Peptide is synthesized with its C-terminus conjugated to 5-[(2-aminoethyl)amino]naphthalene-1-sulfonic acid (EDANS). Casein Kinase 2 Substrate Peptide can be used for protein kinase CK2 activity determination.	price>
R-C-2799	Licofelone (ML3000) CAS:156897-06-2	Licofelone(ML-3000)is a dual COX/5-lipoxygenase(5-LOX)inhibitor(IC50=0.21/0.18μM,respectively) for the treatment of osteoarthritis.Licofelone exerts anti-inflammatory and anti-proliferative effects.Licofelone induces apoptosis,and decreases the production of proinflammatory leukotrienes and prostaglandins.	price>
R-C-3329	DSPE-PEG750-psCPP	(DSPE) polyethyleneglycol is a combination of phospholipid and polyethylene glycol,which has hydrophilicity and hydrophobicity.Polyethylene glycol liposomes were used to form high-quality materials.It can be used for drug delivery,gene transfection and vaccine delivery.Pegylated phospholipids can significantly improve blood circulation time and stabilize drug encapsulation.These materials can also be used for targeted drug delivery by modifying the ligand with the target surface to add antibodies and peptides.	price>
R-R-4499	CK2 inhibitor 2 CAS No.2641079-92-5	CK2 inhibitor 2/CAS No.2641079-92-5 is a potent, selective and orally active inhibitor of CK2, with an IC50 of 0.66 nM. CK2 inhibitor 2 shows high selectivity for Clk2 (IC50=32.69 nM)/CK2. CK2 inhibitor 2 exhibits favorable antiproliferative and antitumor activity.	price>
R-C-2800	GR 103691 CAS:162408-66-4	GR 103691 is a potent,selective dopamine D3 receptor antagonist with a Ki value of 0.4nM.GR 103691 shows more than 100-fold selectivity for human dopamine human(h)D3 over hD4 and hD1 sites.	price>
R-R-4500	Casein kinase 1o-IN-6 CAS No.1579991-01-7	Casein kinase 1δ-IN-6/CAS No.1579991-01-7 is a potent and selective protein kinase CK-1δ inhibitor with an IC50 of 23 nM. Casein kinase 1δ-IN-6 shows neuroprotective and anti-inflammatory properties both in vitro and in vivo. Casein kinase 1δ-IN-6 is a promising drug candidate and can be used for neurodegenerative diseases research.	price>
R-C-2801	ML352 CAS:1649450-12-3	The neurotransmitter acetylcholine(ACh)plays a critical role in autonomic function,motor control,attention,learning, and memory,and reward.ML352 is a novel,noncompetitive inhibitor of the presynaptic choline transporter.	price>
R-R-4501	SRPIN803 CAS No.380572-02-1	SRPIN803/CAS No.380572-02-1 is a potent CK2 and SRPK1 dual inhibitor, with IC50s of 203 nM and 2.4 μM, respectively. SRPIN803 exhibits antiangiogenic activity. SRPIN803 can be used for the research of age-related macular degeneration.	price>

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