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R-R-4359 (Rac)-Razpipadon CAS No.1643462-93-4 PW0464/CAS No.1643462-93-4, a nanomolar potent complete G protein biased ligand, is a noncatechol D1R agonist, with an EC50 of 5.8 nM (Gs-cAMP). price>
R-C-2660 Triapine CAS:200933-27-3 Triapine(3-AP)is a potent ribonucleotide reductase(RNR)inhibitor with broad spectrum antitumor activity by inhibiting DNA synthesis. price>
R-R-4360 MIF-1 TFA CAS No.35240-69-8 MIF-1 TFA (Melanostatin)/CAS No.35240-69-8, an endogenous brain peptide, is a potent dopamine receptor allosteric modulator. MIF-1 TFA inhibits melanin formation. MIF-1 TFA blocks the effects of opioid receptor activation to modulate the analgesic effects. MIF-1 TFA accesses from the blood to the CNS by directly crossing the blood-brain barrier (BBB). price>
R-C-2661 Tasquinimod CAS:254964-60-8 Tasquinimod is an oral antiangiogenic agent,which has the potential for castration-resistant prostate cancer treatment.Tasquinimod binds to the regulatory Zn2+ binding domain of HDAC4 with Kd of 10-30nM.Tasquinimod also is a S100A9 inhibitor. price>
R-R-4361 Alizapride hydrochloride CAS No.59338-87-3 Alizapride/CAS No.59338-87-3 is a potent antiemetic, acting as a dopamine receptor antagonist. Alizapride also used in human digestive disorders. price>
R-C-2662 Paradol CAS:27113-22-0 Paradol is a pungent phenolic substance found in ginger and other Zingiberaceae plants.Paradol is an effective inhibitor of tumor promotion in mouse skin carcinogenesis,binds to cyclooxygenase(COX)-2 active site. price>
R-R-4362 Aramisulpride CAS No.71675-90-6 Aramisulpride/CAS No.71675-90-6 is a dopamine D2 receptor and serotonin receptor antagonist used for the research of metabolic disorders. price>
R-C-2663 XAV-939 CAS:284028-89-3 XAV-939 is a potent tankyrase inhibitor that targets Wnt/β-catenin signaling.XAV-939 stabilizes axin by inhibiting tankyrase 1 and tankyrase 2(IC50s of 5 and 2nM,respectively),thereby stimulating β-catenin degradation.XAV939 binds tightly to the catalytic(PARP)domains of TNKS1 and TNKS2(Kds of 99 and 93nM,respectively). price>
R-R-4363 (R)-Preclamol hydrochloride CAS No.89874-80-6 (R)-Preclamol hydrochloride ((+)-3-PPP hydrochloride)/CAS No.89874-80-6 is the R-enantiomer of Preclamol hydrochloride. (R)-Preclamol hydrochloride is a DA agonist with autoreceptor as well as postsynaptic receptor stimulatory properties. price>
R-C-2664 Teniposide CAS:29767-20-2 Teniposide(NSC 122819,VM-26)is a chemotherapeutic medication mainly used in the treatment of childhood acute lymphocytic leukemia(ALL). price>
R-R-4364 Medifoxamine CAS No.32359-34-5 Medifoxamine/CAS No.32359-34-5 is a monoamine re-uptake inhibiting antidepressive agent which preferentially inhibits dopamine reuptake. price>
R-C-2665 Zidovudine CAS:30516-87-1 Zidovudine is a nucleoside analog reverse-transcriptase inhibitor(NRTI),a type of antiretroviral drug used for the treatment of HIV/AIDS infection.Azidothymidine decreases CRISPR-mediated homology directed repair(HDR)efficiency. price>
R-R-4365 Zuclopenthixol dihydrochloride CAS No.58045-23-1 Zuclopenthixol ((Z)-Clopenthixol) dihydrochloride/CAS No.58045-23-1 is a thioxanthene derivative which acts as a mixed dopamine D1/D2 receptor antagonist. Zuclopenthixol dihydrochloride is used in the study of schizophrenia. price>
R-C-2666 Palifosfamide CAS:31645-39-3 Palifosfamide is a novel DNA alkylator and the active metabolite of ifosfamide, with antitumor activity. price>
R-R-4366 Haloperidol-d4 CAS No.1189986-59-1 Haloperidol-d4/CAS No.1189986-59-1 is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist. price>
R-C-2567 Z-YVAD-FMK CAS:210344-97-1 Z-YVAD-FMK is a cell-permeable caspase-1 and -4 inhibitor with anti-inflammatory and anti-tumor activities. price>
R-C-2667 BIBR 1532 CAS:321674-73-1 BIBR1532 is a selective telomerase inhibitor.BIBR1132 is highly selective for inhibition of telomerase,resulting in delayed growth arrest of tumor cells. price>
R-C-2687 KD 5170 CAS:940943-37-3 KD 5170,a novel mercaptoketone-based histone deacetylase inhibitor that exhibits broad spectrum antitumor activity in vitro and in vivo. price>
R-R-4367 (-)-GSK598809 hydrochloride CAS No.863766-31-8 (-)-GSK598809/CAS No.863766-31-8 is an isomer of GSK598809. GSK598809 is a potent and selective dopamine D3 Receptor (DRD3) antagonist. price>
R-C-2568 Zotiraciclib CAS:1204918-72-8 Zotiraciclib(TG02;SB1317)is a potent inhibitor of CDK2,JAK2,and FLT3 for the treatment of cancer,with IC50s of 13,73,and 56 nM for CDK2,JAK2 and FLT3,respectively. price>