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Catalog	name	Description	price
R-R-4497	PI-828 CAS No.942289-87-4	PI-828/CAS No.942289-87-4 is a dual PI3K and casein kinase 2 (CK2) inhibitor with IC50s of 173 nM, 149 nM, and 1127 nM for p110α, CK2, and CK2α2 in lipid kinase assay, respectively.	price>
R-C-2798	Pizotifen CAS:15574-96-6	Pizotifen is a serotonin antagonist which acts mainly at the 5-HT1,5-HT2A,and 5HT2C receptors with some antihistamine activity.	price>
R-C-3328	DSPE-PEG550-psCPP	(DSPE) polyethyleneglycol is a combination of phospholipid and polyethylene glycol,which has hydrophilicity and hydrophobicity.Polyethylene glycol liposomes were used to form high-quality materials.It can be used for drug delivery,gene transfection and vaccine delivery.Pegylated phospholipids can significantly improve blood circulation time and stabilize drug encapsulation.These materials can also be used for targeted drug delivery by modifying the ligand with the target surface to add antibodies and peptides.	price>
R-R-4498	Casein Kinase 2 Substrate Peptide CAS No.132176-35-3	Casein Kinase 2 Substrate Peptide is a common CK2 substrate peptide. Casein Kinase 2 Substrate Peptide is synthesized with its C-terminus conjugated to 5-[(2-aminoethyl)amino]naphthalene-1-sulfonic acid (EDANS). Casein Kinase 2 Substrate Peptide can be used for protein kinase CK2 activity determination.	price>
R-C-2799	Licofelone (ML3000) CAS:156897-06-2	Licofelone(ML-3000)is a dual COX/5-lipoxygenase(5-LOX)inhibitor(IC50=0.21/0.18μM,respectively) for the treatment of osteoarthritis.Licofelone exerts anti-inflammatory and anti-proliferative effects.Licofelone induces apoptosis,and decreases the production of proinflammatory leukotrienes and prostaglandins.	price>
R-C-3329	DSPE-PEG750-psCPP	(DSPE) polyethyleneglycol is a combination of phospholipid and polyethylene glycol,which has hydrophilicity and hydrophobicity.Polyethylene glycol liposomes were used to form high-quality materials.It can be used for drug delivery,gene transfection and vaccine delivery.Pegylated phospholipids can significantly improve blood circulation time and stabilize drug encapsulation.These materials can also be used for targeted drug delivery by modifying the ligand with the target surface to add antibodies and peptides.	price>
R-R-4499	CK2 inhibitor 2 CAS No.2641079-92-5	CK2 inhibitor 2/CAS No.2641079-92-5 is a potent, selective and orally active inhibitor of CK2, with an IC50 of 0.66 nM. CK2 inhibitor 2 shows high selectivity for Clk2 (IC50=32.69 nM)/CK2. CK2 inhibitor 2 exhibits favorable antiproliferative and antitumor activity.	price>
R-C-2800	GR 103691 CAS:162408-66-4	GR 103691 is a potent,selective dopamine D3 receptor antagonist with a Ki value of 0.4nM.GR 103691 shows more than 100-fold selectivity for human dopamine human(h)D3 over hD4 and hD1 sites.	price>
R-R-4500	Casein kinase 1o-IN-6 CAS No.1579991-01-7	Casein kinase 1δ-IN-6/CAS No.1579991-01-7 is a potent and selective protein kinase CK-1δ inhibitor with an IC50 of 23 nM. Casein kinase 1δ-IN-6 shows neuroprotective and anti-inflammatory properties both in vitro and in vivo. Casein kinase 1δ-IN-6 is a promising drug candidate and can be used for neurodegenerative diseases research.	price>
R-C-2801	ML352 CAS:1649450-12-3	The neurotransmitter acetylcholine(ACh)plays a critical role in autonomic function,motor control,attention,learning, and memory,and reward.ML352 is a novel,noncompetitive inhibitor of the presynaptic choline transporter.	price>
R-R-4501	SRPIN803 CAS No.380572-02-1	SRPIN803/CAS No.380572-02-1 is a potent CK2 and SRPK1 dual inhibitor, with IC50s of 203 nM and 2.4 μM, respectively. SRPIN803 exhibits antiangiogenic activity. SRPIN803 can be used for the research of age-related macular degeneration.	price>
R-C-2802	MSPG CAS:169209-64-7	Relatively non-selective antagonist of presynaptic mGlu receptors in neonatal rat spinal cord and adult rat cerebrocortical mGlu receptors.	price>
R-R-4502	Casein kinase 1o-IN-8 CAS No.851396-73-1	Casein kinase 1δ-IN-8 (compound 494)/CAS No.851396-73-1 is an inhibitor of Casein kinase 1δ, Casein kinase 1δ-IN-8 can be used in the treatment of neurodegenerative disorders such as Alzheimer disease.	price>
R-C-2803	MTPG CAS:169209-66-9	MTPG is a group II/group III mGlu antagonist,showing selectivity for group II in electrophysiological studies.MTPG is a potent antagonist for(1S,3S)-ACPD-sensitive receptors;preference for group II mGluR.	price>
R-R-4503	Casein kinase 1o-IN-1 CAS No.851871-94-8	Casein kinase 1δ-IN-1 (compound 822)/CAS No.851871-94-8 is an inhibitor of casein kinase 1 delta (CK1δ), exhibits inhibition of greater than 5%. Casein kinase 1δ-IN-1 can be used for neurodegenerative disorders such as Alzheimer disease research.	price>
R-C-2804	Eglumegad (LY354740) CAS:176199-48-7	Eglumegad(LY354740)is a highly potent and selective group II(mGlu2/3)receptor agonist with IC50s of 5 and 24nM on transfected human mGlu2 and mGlu3 receptors,respectively.	price>
R-R-4504	ON 108600 CAS No.1585246-23-6	ON 108600/CAS No.1585246-23-6 is a inhibitor for CK2 (Casein Kinase2)/TNIK/DYRK1 , with the IC50s for DYRK1A/DYRKB, DYRK2, CK2α1/CK2α2, and TNIK of 0.016 μm/0.007 μM, 0.028 μM, 0.05 μM/0.005 μM, and 0.005 μM, respectively. ON 108600 has antitumor activity.	price>
R-C-2805	NKP608 CAS:177707-12-9	NKP608 is a non-peptidic derivative of 4-aminopiperidine which acts as a selective,specific and potent antagonist at the neurokinin-1(NK-1)receptor both in vitro(IC50=2.6nM)and in vivo.	price>
R-R-4505	Casein kinase 1o-IN-9 CAS No.854355-54-7	Casein kinase 1δ-IN-9 (compound 737)/CAS No.854355-54-7 is a potent casein kinase 1δ (CK1δ/CK15) inhibitor. Casein kinase 1δ-IN-9 can be used for the research of neurodegenerative disorders such as Alzheimer disease.	price>
R-C-2806	Sumanirole maleate CAS:179386-44-8	Sumanirole maleate(U-95666E;PNU-95666E)is a highly selective D2 receptor full agonist with an ED50 of about 46nM.Sumanirole was developed for the treatment of Parkinson is disease and restless leg syndrome.	price>

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