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Catalog | name | Description | price |
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R-R-4366 | Haloperidol-d4 CAS No.1189986-59-1 | Haloperidol-d4/CAS No.1189986-59-1 is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist. | price> |
R-C-2567 | Z-YVAD-FMK CAS:210344-97-1 | Z-YVAD-FMK is a cell-permeable caspase-1 and -4 inhibitor with anti-inflammatory and anti-tumor activities. | price> |
R-C-2667 | BIBR 1532 CAS:321674-73-1 | BIBR1532 is a selective telomerase inhibitor.BIBR1132 is highly selective for inhibition of telomerase,resulting in delayed growth arrest of tumor cells. | price> |
R-C-2687 | KD 5170 CAS:940943-37-3 | KD 5170,a novel mercaptoketone-based histone deacetylase inhibitor that exhibits broad spectrum antitumor activity in vitro and in vivo. | price> |
R-R-4367 | (-)-GSK598809 hydrochloride CAS No.863766-31-8 | (-)-GSK598809/CAS No.863766-31-8 is an isomer of GSK598809. GSK598809 is a potent and selective dopamine D3 Receptor (DRD3) antagonist. | price> |
R-C-2568 | Zotiraciclib CAS:1204918-72-8 | Zotiraciclib(TG02;SB1317)is a potent inhibitor of CDK2,JAK2,and FLT3 for the treatment of cancer,with IC50s of 13,73,and 56 nM for CDK2,JAK2 and FLT3,respectively. | price> |
R-C-2668 | AG-14361 CAS:328543-09-5 | AG14361 is a potent PARP-1 inhibitor,with a Ki of < 5nM,and in permeabilized SW620 and intact SW620 cells,the IC50s are 29nM and 14nM,respectively. | price> |
R-C-2688 | TCS HDAC6 20b CAS:956154-63-5 | TCS HDAC6 20b,selective inhibitor of histone deacetylase 6(HDAC6).Inhibits HCT116 growth in combination with taxol. Also inhibits growth of MCF-7 cells stimulated by estrogen. | price> |
R-R-4368 | Ro 10-5824 dihydrochloride CAS No.189744-94-3 | Ro 10-5824 dihydrochloride/CAS No.189744-94-3 is a selective dopamine D4 receptor partial agonist, with Ki of 5.2 nM. | price> |
R-C-2569 | Zotepine CAS:26615-21-4 | Zotepine,an antipsychotic agent,is a potent antagonist of 5-HT2A,5-HT2C,Histamine H1,α1-adrenergic and Dopamine D2 receptors,with Kds of 2.6nM,3.2nM,3.3nM,7.3nM and 8nM,respectively.Zotepine exhibits antidepressive and anxiolytic effects in vivo. | price> |
R-C-2669 | Viomycin CAS:32988-50-4 | Viomycin(free base)is a tuberactinomycin antibiotic essential for treating multidrug-resistant tuberculosis.It inhibits bacterial protein synthesis by blocking elongation factor G(EF-G)catalyzed translocation of messenger RNA on the ribosome. | price> |
R-R-4369 | Pentiapine CAS No.81382-51-6 | Pentiapine (CGS 10746)/CAS No.81382-51-6 is a dopamine release inhibitor without binding to synaptic dopamine receptor sites. | price> |
R-C-2670 | NSC 3852 CAS:3565-26-2 | NSC 3852 is an HDAC(histone deacetylase)inhibitor. | price> |
R-R-4370 | NMI 8739 CAS No.129024-87-9 | NMI 8739/CAS No.129024-87-9 is a dopamine D2 autoreceptor agonist, which is an amine conjugate of the DHA carrier and the neurotransmitter dopamine. | price> |
R-C-2671 | Penciclovir CAS:39809-25-1 | Penciclovir is reported to be potent against HSV types 1 and 2 with IC50 of 0.04-1.8μg/mL and 0.06-4.4μg/mL,respectively. | price> |
R-R-4371 | L-DOPA-d6 CAS No.713140-75-1 | L-DOPA-d6/CAS No.713140-75-1 is the deuterium labeled L-DOPA. L-DOPA (Levodopa) is an orally active metabolic precursor of neurotransmitters dopamine. L-DOPA can cross the blood-brain barrier and is converted into dopamine in the brain. | price> |
R-C-2672 | Flumequine CAS:42835-25-6 | Flumequine(R-802)is a quinolone antibiotic,and acts as a topoisomerase II inhibitor,with an IC50 of 15μM(3.92μg/mL). | price> |
R-R-4372 | Odapipam CAS No.131796-63-9 | Odapipam (NNC 756)/CAS No.131796-63-9 is a selective, high affinity and benzazepine dopamine D1 receptor antagonist with a Kd of 0.18 nM. Odapipam is also a superior positron emission tomography (PET) radiotracer. | price> |
R-C-2673 | Beta-Lapachone CAS:4707-32-8 | Beta-Lapachone is a selective DNA topoisomerase I inhibitor,exhibiting no inhibitory activities against DNA topoisomerase II or ligase. | price> |
R-R-4373 | Preclamol hydrochloride CAS No.88768-67-6 | Preclamol hydrochloride ((-)-3-PPP hydrochloride)/CAS No.88768-67-6 is a selective dopamine autoreceptor agonist. Preclamol hydrochloride has the potential for the research of schizophrenia. | price> |