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Catalog | name | Description | price |
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R-R-4356 | Bacopaside X CAS No.94443-88-6 | Bacopaside X/CAS No.94443-88-6 is found in Bacopa monnieri, and shows a binding affinity toward the D1 receptor. | price> |
R-C-2657 | Dp44mT CAS: 152095-12-0 | Dp44mT is an iron chelator,possessing DNA-damaging activity mediated by top2a inhibition. | price> |
R-R-4357 | Naxagolide CAS No.88058-88-2 | Naxagolide ((+)-PHNO; Dopazinol)/CAS No.88058-88-2 is a potent dopamine D2 (Dopamine Receptor) agonist. Naxagolide has the potential for the research of parkinson disease (PD). | price> |
R-C-2658 | SCH 51344 CAS:171927-40-5 | SCH-51344 is an inhibitor of RAS/RAC-mediated cell morphology pathway.RAS interacts with multiple targets in the cell and controls at least two signaling pathways,one regulating extracellular signal-regulated kinase(ERK)activation and the other controlling membrane ruffling formation. | price> |
R-R-4358 | JNJ-37822681 dihydrochloride CAS No.2108806-02-4 | JNJ-37822681 dihydrochloride/CAS No.2108806-02-4 is a potent, specific, centrally active, fast-dissociating dopamine D2 receptor antagonist with a moderate binding affinity for the dopamine D2L receptor (Ki =158 nM), which has potential for the treatment of schizophrenia and bipolar disorder. | price> |
R-C-2659 | Apicidin CAS:183506-66-3 | Apicidin(OSI 2040)is a fungal metabolite, acts as a histone deacetylase(HDAC)inhibitor,with antiparasitic activity and a broad spectrum antiproliferative activity. | price> |
R-R-4359 | (Rac)-Razpipadon CAS No.1643462-93-4 | PW0464/CAS No.1643462-93-4, a nanomolar potent complete G protein biased ligand, is a noncatechol D1R agonist, with an EC50 of 5.8 nM (Gs-cAMP). | price> |
R-C-2660 | Triapine CAS:200933-27-3 | Triapine(3-AP)is a potent ribonucleotide reductase(RNR)inhibitor with broad spectrum antitumor activity by inhibiting DNA synthesis. | price> |
R-R-4360 | MIF-1 TFA CAS No.35240-69-8 | MIF-1 TFA (Melanostatin)/CAS No.35240-69-8, an endogenous brain peptide, is a potent dopamine receptor allosteric modulator. MIF-1 TFA inhibits melanin formation. MIF-1 TFA blocks the effects of opioid receptor activation to modulate the analgesic effects. MIF-1 TFA accesses from the blood to the CNS by directly crossing the blood-brain barrier (BBB). | price> |
R-C-2661 | Tasquinimod CAS:254964-60-8 | Tasquinimod is an oral antiangiogenic agent,which has the potential for castration-resistant prostate cancer treatment.Tasquinimod binds to the regulatory Zn2+ binding domain of HDAC4 with Kd of 10-30nM.Tasquinimod also is a S100A9 inhibitor. | price> |
R-R-4361 | Alizapride hydrochloride CAS No.59338-87-3 | Alizapride/CAS No.59338-87-3 is a potent antiemetic, acting as a dopamine receptor antagonist. Alizapride also used in human digestive disorders. | price> |
R-C-2662 | Paradol CAS:27113-22-0 | Paradol is a pungent phenolic substance found in ginger and other Zingiberaceae plants.Paradol is an effective inhibitor of tumor promotion in mouse skin carcinogenesis,binds to cyclooxygenase(COX)-2 active site. | price> |
R-R-4362 | Aramisulpride CAS No.71675-90-6 | Aramisulpride/CAS No.71675-90-6 is a dopamine D2 receptor and serotonin receptor antagonist used for the research of metabolic disorders. | price> |
R-C-2663 | XAV-939 CAS:284028-89-3 | XAV-939 is a potent tankyrase inhibitor that targets Wnt/β-catenin signaling.XAV-939 stabilizes axin by inhibiting tankyrase 1 and tankyrase 2(IC50s of 5 and 2nM,respectively),thereby stimulating β-catenin degradation.XAV939 binds tightly to the catalytic(PARP)domains of TNKS1 and TNKS2(Kds of 99 and 93nM,respectively). | price> |
R-R-4363 | (R)-Preclamol hydrochloride CAS No.89874-80-6 | (R)-Preclamol hydrochloride ((+)-3-PPP hydrochloride)/CAS No.89874-80-6 is the R-enantiomer of Preclamol hydrochloride. (R)-Preclamol hydrochloride is a DA agonist with autoreceptor as well as postsynaptic receptor stimulatory properties. | price> |
R-C-2664 | Teniposide CAS:29767-20-2 | Teniposide(NSC 122819,VM-26)is a chemotherapeutic medication mainly used in the treatment of childhood acute lymphocytic leukemia(ALL). | price> |
R-R-4364 | Medifoxamine CAS No.32359-34-5 | Medifoxamine/CAS No.32359-34-5 is a monoamine re-uptake inhibiting antidepressive agent which preferentially inhibits dopamine reuptake. | price> |
R-C-2665 | Zidovudine CAS:30516-87-1 | Zidovudine is a nucleoside analog reverse-transcriptase inhibitor(NRTI),a type of antiretroviral drug used for the treatment of HIV/AIDS infection.Azidothymidine decreases CRISPR-mediated homology directed repair(HDR)efficiency. | price> |
R-R-4365 | Zuclopenthixol dihydrochloride CAS No.58045-23-1 | Zuclopenthixol ((Z)-Clopenthixol) dihydrochloride/CAS No.58045-23-1 is a thioxanthene derivative which acts as a mixed dopamine D1/D2 receptor antagonist. Zuclopenthixol dihydrochloride is used in the study of schizophrenia. | price> |
R-C-2666 | Palifosfamide CAS:31645-39-3 | Palifosfamide is a novel DNA alkylator and the active metabolite of ifosfamide, with antitumor activity. | price> |