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Catalog	name	Description	price
R-R-4389	FAUC 365 CAS No.474432-66-1	FAUC 365/CAS No.474432-66-1 is a highly dopamine D3 receptor-selective antagonist with Ki values of 0.5 nM, 340, 2600, and 3600 nM at D3, D4.4, D2short, and D2Long receptors, respectively. FAUC 365 can be used for the research of schizophrenia, and Parkinson disease.	price>
R-C-2690	SGI-1027 CAS：1020149-73-8	SGI-1027 is a DNA methyltransferase(DNMT)inhibitor,with IC50s of 7.5μM,8μM, and 12.5 μM for DNMT3B,DNMT3A,and DNMT1 with poly(dI-dC)as substrate.	price>
R-R-4390	SK609 hydrochloride CAS No.1092797-77-7	SK609 hydrochloride/CAS No.1092797-77-7 is a dopamine D3 receptor (D3R) selective agonist with an EC50 of 1109 nM. SK609 hydrochloride has the potential for parkinson research.	price>
R-C-2691	LB-100 CAS：1026680-07-8	LB-100 is a protein phosphatase 2A(PP2A)inhibitor.LB-100 sensitizes hepatocellular carcinoma cells to the effects of sorafenib during hypoxia by activation of Smad3 phosphorylation.LB-100 enhanced the effects of sorafenib in HCC cells only during hypoxic environments.	price>
R-R-4391	Levosulpiride-d3 CAS No.124020-27-5	Levosulpiride-d3/CAS No.124020-27-5 is the deuterium labeled Levosulpiride. Levosulpiride (RV-12309) is the (S)-enantiomer of sulpiride, which is a D2 receptor a antagonist, an atypical antipsychotic agent of the benzamide class.	price>
R-C-2692	NVP-BSK805 CAS：1092499-93-8	NVP-BSK805 is a JAK2 inhibor,which displays more than 20-fold selectivity towards JAK2 in vitro,as well as excellent selectivity in broader kinase profiling.In vivo,NVP-BSK805 exhibited good oral bioavailability and a long half-life.	price>
R-R-4392	CP 226269 CAS No.220941-93-5	CP 226269/CAS No.220941-93-5 is a potent dopamine D4 receptor agonist that induces calcium flux with EC50 of 32.0 nM. CP 226269 can be used in the research of schizophrenia and other related diseases.	price>
R-C-2693	CCT137690 CAS：1095382-05-0	CCT 137690 is a potent and orally available aurora kinase inhibitor with IC50s of 15,25,and 19nM for aurora A,B and C,respectively.	price>
R-R-4393	FAUC 213 CAS No.337972-47-1	FAUC 213/CAS No.337972-47-1 is an orally active and highly selective dopamine D4 receptor complete antagonist with a Ki of 2.2 nM for hD4.4. FAUC 213 has less activity on D2 and D3 receptors (Kis of 3.4 μM, 5.3 μM for hD2, hD3, respectively). FAUC 213 can cross the blood-brain barrier (BBB). FAUC 213 exhibits atypical antipsychotic characteristic.	price>
R-C-2694	BYK 204165 CAS：1104546-89-5	BYK204165 is a potent and selective PARP1 inhibitor. BYK204165 inhibits cell-free recombinant human PARP-1(hPARP-1)with a pIC50 of 7.35(pKi=7.05),and murine PARP-2(mPARP-2)with a pIC50 of 5.38,respectively.BYK204165 displays 100-fold selectivity for PARP-1.	price>
R-R-4394	BP 897 hydrochloride CAS No.314776-92-6	BP 897 hydrochloride/CAS No.314776-92-6 is a potent and partial dopamine D3 receptor agonist and a weak D2 receptor antagonist. BP 897 hydrochloride displays a high affinity at the dopamine D3 receptor (Ki=0.92 nM) and a 70 times lower affinity at the D2 receptor (Ki=61 nM).	price>
R-C-2695	Lestaurtinib CAS：111358-88-4	Lestaurtinib(CEP-701;KT-5555)is a multi-kinase inhibitor with potent activity against the Trk family of receptor tyrosine kinases.Lestaurtinib inhibits JAK2, FLT3 and TrkA with IC50s of 0.9,3 and less than 25nM,respectively.	price>
R-R-4395	FAUC 346 CAS No.474432-65-0	FAUC 346/CAS No.474432-65-0, a highly selective D3 partial agonist (EC50 = 1.5 nM).	price>
R-C-2696	MCB-613 CAS：1162656-22-5	MCB-613 is a potent Steroid Receptor Coactivator Stimulator that Overstimulates Cancer Cells and Leads to Cell Stress and Death.MCB-613 can super-stimulate SRCs transcriptional activity.MCB-613 increases SRCs interactions with other coactivators and markedly induces ER stress coupled to the generation of reactive oxygen species(ROS).	price>
R-R-4396	Bromperidol (Standard) CAS No.10457-90-6	Bromperidol (Standard)/CAS No.10457-90-6 is the analytical standard of Bromperidol. This product is intended for research and analytical applications. Bromperidol (R-11333) possesses antipsychotic activity, with a high affinity for central dopamine receptors D2. Bromperidol can kill Mycobacteria in a synergistic manner with Spectinomycin.	price>
R-C-2697	UNC 0224 CAS：1197196-48-7	UNC0224 is a potent and selective histone methyltransferase G9a inhibitor with a Ki of 2.6nM,an IC50 of 15nM and a Kd of 23nM.UNC0224 also potently inhibits b>GLP with assay-dependent IC50 values of 20-58nM.	price>
R-R-4397	L-DOPA-13C CAS No.586971-29-1	L-DOPA-13C/CAS No.586971-29-1 is the 13C labeled L-DOPA[1]. L-DOPA (Levodopa) is an orally active metabolic precursor of neurotransmitters dopamine. L-DOPA can cross the blood-brain barrier and is converted into dopamine in the brain.	price>
R-C-2698	Tautomycetin CAS：119757-73-2	Tautomycetin is a potent and specifical PP1 inhibitor with the potential apoptosis-inducing activity.Tautomycetin inhibits purified PP1 and PP2A enzymes with IC50s of 1.6nM and 62nM,respectively.Tautomycetin is an antifungal antibiotic and has immunosuppressive effects in vivo.	price>
R-R-4398	Asimilobine CAS No.6871-21-2	Asimilobine/CAS No.6871-21-2 is an aporphine isoquinoline alkaloid isolated from plant species of Magnolia obobata Thun. Asimilobine is a dopamine biosynthesis inhibitor and a serotonergic receptor antagonist. Asimilobine shows an antimalarial and anti-cancer activity.	price>
R-C-2699	AZD1208 CAS：1204144-28-4	AZD1208 is orally available,small molecule inhibitor of PIM kinases with potential antineoplastic activity.Pan-PIM kinase inhibitor AZD1208 inhibits the activities of PIM1,PIM2 and PIM3 serine/threonine kinases,which may result in the interruption of the G1/S phase cell cycle transition,thereby causing cell cycle arrest and inducing apoptosis in cells that overexpress PIMs.	price>

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