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Catalog	name	Description	price
R-R-4297	Sulpiride CAS No.15676-16-1	Sulpiride/CAS No.15676-16-1 is an orally active dopamine D2/D3 receptor antagonist. Sulpiride is an atypical antipsychotic agent of the benzamide family. Sulpiride can be used in research into anxiety, depression and breast cancer.	price>
R-C-2598	Matrine CAS:519-02-8	Matrine,a novel autophagy inhibitor,possesses anti-inflammation, immunosuppression,anti-fibrotic and anticancer activities,it could inhibit cell proliferation and induce apoptosis of SGC-7901 cells in vitro by up-regulating Fas/FasL expression and activating caspase-3 enzyme.	price>
R-R-4298	Raclopride CAS No.84225-95-6	Raclopride/CAS No.84225-95-6 is a dopamine D2/D3 receptor antagonist with potential antipsychotic effects. Raclopride binds to D2 and D3 receptors with Kis of 1.8 nM and 3.5 nM, respectively.	price>
R-C-2599	Embelin CAS:550-24-3	Embelin(Embelic acid),a potent,nonpeptidic XIAP inhibitor(IC50=4.1μM), inhibits cell growth,induces apoptosis, and activates caspase-9 in prostate cancer cells with high levels of XIAP.Embelin blocks NF-kappaB signaling pathway leading to suppression of NF-kappaB-regulated antiapoptotic and metastatic gene products.	price>
R-R-4299	SKF-82958 hydrobromide CAS No.74115-01-8	SKF-82958 ((±)-SKF 82958) hydrobromide/CAS No.74115-01-8 is a dopamine D1 receptor full agonist (K0.5=4 nM), displays selective for D1 over D2 receptors (K0.5=73 nM). SKF-82958 hydrobromide induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striatal membranes (EC50=491 nM).	price>
R-C-2600	NSC 66811 CAS:6964-62-1	NSC 66811 is a MDM2-p53 inhibitor,with a Ki of 120nM for binding to MDM2.	price>
R-R-4300	Dihydrexidine hydrochloride CAS No.137417-08-4	Dihydrexidine hydrochloride (DAR-0100 hydrochloride)/CAS No.137417-08-4 is a high potent, selective and full efficacy D1-like dopamine receptor (D1/D5) agonist, with an IC50 of 10 nM for D1 receptor. Dihydrexidine hydrochloride exhibits potent antiparkinsonian activity. Dihydrexidine hydrochloride can stimulate YAP phosphorylation.	price>
R-C-2601	Mcl1-IN-1 CAS:713492-66-1	Mcl1-IN-1 is a potent and selective inhibitor of the apoptosis regulating proteins Mcl-1.	price>
R-R-4301	Tetrahydropalmatine CAS No.2934-97-6	Tetrahydropalmatine/CAS No.2934-97-6 possesses analgesic effects. Tetrahydropalmatine acts through inhibition of amygdaloid release of dopamine to inhibit an epileptic attack in rats.	price>
R-C-2602	NSC 319726 CAS:71555-25-4	NSC319726(ZMC1)is a mutant p53R175 reactivator;inhibits growth of fibroblasts expressing the p53R175 mutation(IC50=8nM);shows no inhibition for p53 wild-type cells.	price>
R-R-4302	Pergolide mesylate CAS No.66104-23-2	Pergolide mesylate (Pergolide methanesulfonate)/CAS No.66104-23-2, an Ergoline derivative, is a potent and orally active dopamine D1 and D2 receptors agonist.	price>
R-C-2603	MIRA-1NSC19630 CAS:72835-26-8	MIRA-1 restores wild-type conformation,function and DNA binding activity to mutant p53.Induces p53 transcriptional transactivation of p21,MDM2 and PUMA.	price>
R-R-4303	Tetrahydroberberine CAS No.522-97-4	Tetrahydroberberine/CAS No.522-97-4 is a different kind of living thing that can be extended and divided into parts. Tetrahydroberberine is a kind of effective D2 receptor antagonistic force. Tetrahydroberberine has the ability to strengthen the stomach and relieve the pressure on the stomach.	price>
R-C-2604	Brassinolide CAS:72962-43-7	Brassinolide,a plant steroid isolated from Brassica napus pollen,promotes cell elongation and cell devision and thus regulates plant growth and development.	price>
R-R-4304	Ralmitaront CAS No.2133417-13-5	Ralmitaront (RO6889450)/CAS No.2133417-13-5 is an orally active agonist of trace amine-associated receptor 1 (TAAR1) with a EC50 value of 110.4 nM. Ralmitaront has antipsychotic, cognitively improvement, and antidepressant activity in rodents. Ralmitaront can be used as a neurosuppressant in the study of neuro-related diseases, such as schizophrenia (SCZ), schizoaffective disorder.	price>
R-C-2605	Ivachtin CAS:745046-84-8	Ivachtin(Caspase-3 Inhibitor VII;compound 7a)is a nonpeptide,noncompetitive and reversibl caspase-3 inhibitor with an IC50 of 23nM.Ivachtin has modest selectivity for the remaining caspases.	price>
R-R-4305	Ropinirole hydrochloride CAS No.91374-20-8	Ropinirole (SKF 101468) hydrochloride/CAS No.91374-20-8 is an orally active, potent D3/D2 receptor agonist with a Ki of 29 nM for D2 receptor. Ropinirole hydrochloride has pEC50s of 7.4, 8.4 and 6.8 for hD2, hD3 and hD4 receptors, respectively. Ropinirole hydrochloride has no affinity for the D1 receptors.	price>
R-C-2606	Epibrassinolide CAS:78821-43-9	Epibrassinolide(24-Epibrassinolide)is a ubiquitously occurring plant growth hormone which shows great potential to alleviate heavy metals and pesticide stress in plants.Epibrassinolide is a potential apoptotic inducer in various cancer cells without affecting the non-tumor cell growth.	price>
R-R-4306	Pramipexole dihydrochloride CAS No.104632-25-9	Pramipexole dihydrochloride/CAS No.104632-25-9 is a selective and blood-brain barrier (BBB) penetrant dopamine D2-type receptor agonist, with Kis of 2.2 nM, 3.9 nM, 0.5 nM and 1.3 nM for D2-type receptor, D2, D3 and D4 receptors, respectively.	price>
R-C-2607	Roquinimex CAS:84088-42-6	Roquinimex(Linomide;PNU212616;ABR212616)is a quinoline derivative immunostimulant which increases NK cell activity and macrophage cytotoxicity; inhibits angiogenesis and reduces the secretion of TNF alpha.	price>

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