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Catalog | name | Description | price |
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R-C-2661 | Tasquinimod CAS:254964-60-8 | Tasquinimod is an oral antiangiogenic agent,which has the potential for castration-resistant prostate cancer treatment.Tasquinimod binds to the regulatory Zn2+ binding domain of HDAC4 with Kd of 10-30nM.Tasquinimod also is a S100A9 inhibitor. | price> |
R-R-4361 | Alizapride hydrochloride CAS No.59338-87-3 | Alizapride/CAS No.59338-87-3 is a potent antiemetic, acting as a dopamine receptor antagonist. Alizapride also used in human digestive disorders. | price> |
R-C-2662 | Paradol CAS:27113-22-0 | Paradol is a pungent phenolic substance found in ginger and other Zingiberaceae plants.Paradol is an effective inhibitor of tumor promotion in mouse skin carcinogenesis,binds to cyclooxygenase(COX)-2 active site. | price> |
R-R-4362 | Aramisulpride CAS No.71675-90-6 | Aramisulpride/CAS No.71675-90-6 is a dopamine D2 receptor and serotonin receptor antagonist used for the research of metabolic disorders. | price> |
R-C-2663 | XAV-939 CAS:284028-89-3 | XAV-939 is a potent tankyrase inhibitor that targets Wnt/β-catenin signaling.XAV-939 stabilizes axin by inhibiting tankyrase 1 and tankyrase 2(IC50s of 5 and 2nM,respectively),thereby stimulating β-catenin degradation.XAV939 binds tightly to the catalytic(PARP)domains of TNKS1 and TNKS2(Kds of 99 and 93nM,respectively). | price> |
R-R-4363 | (R)-Preclamol hydrochloride CAS No.89874-80-6 | (R)-Preclamol hydrochloride ((+)-3-PPP hydrochloride)/CAS No.89874-80-6 is the R-enantiomer of Preclamol hydrochloride. (R)-Preclamol hydrochloride is a DA agonist with autoreceptor as well as postsynaptic receptor stimulatory properties. | price> |
R-C-2664 | Teniposide CAS:29767-20-2 | Teniposide(NSC 122819,VM-26)is a chemotherapeutic medication mainly used in the treatment of childhood acute lymphocytic leukemia(ALL). | price> |
R-R-4364 | Medifoxamine CAS No.32359-34-5 | Medifoxamine/CAS No.32359-34-5 is a monoamine re-uptake inhibiting antidepressive agent which preferentially inhibits dopamine reuptake. | price> |
R-C-2665 | Zidovudine CAS:30516-87-1 | Zidovudine is a nucleoside analog reverse-transcriptase inhibitor(NRTI),a type of antiretroviral drug used for the treatment of HIV/AIDS infection.Azidothymidine decreases CRISPR-mediated homology directed repair(HDR)efficiency. | price> |
R-R-4365 | Zuclopenthixol dihydrochloride CAS No.58045-23-1 | Zuclopenthixol ((Z)-Clopenthixol) dihydrochloride/CAS No.58045-23-1 is a thioxanthene derivative which acts as a mixed dopamine D1/D2 receptor antagonist. Zuclopenthixol dihydrochloride is used in the study of schizophrenia. | price> |
R-C-2666 | Palifosfamide CAS:31645-39-3 | Palifosfamide is a novel DNA alkylator and the active metabolite of ifosfamide, with antitumor activity. | price> |
R-R-4366 | Haloperidol-d4 CAS No.1189986-59-1 | Haloperidol-d4/CAS No.1189986-59-1 is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist. | price> |
R-C-2567 | Z-YVAD-FMK CAS:210344-97-1 | Z-YVAD-FMK is a cell-permeable caspase-1 and -4 inhibitor with anti-inflammatory and anti-tumor activities. | price> |
R-C-2667 | BIBR 1532 CAS:321674-73-1 | BIBR1532 is a selective telomerase inhibitor.BIBR1132 is highly selective for inhibition of telomerase,resulting in delayed growth arrest of tumor cells. | price> |
R-C-2687 | KD 5170 CAS:940943-37-3 | KD 5170,a novel mercaptoketone-based histone deacetylase inhibitor that exhibits broad spectrum antitumor activity in vitro and in vivo. | price> |
R-R-4367 | (-)-GSK598809 hydrochloride CAS No.863766-31-8 | (-)-GSK598809/CAS No.863766-31-8 is an isomer of GSK598809. GSK598809 is a potent and selective dopamine D3 Receptor (DRD3) antagonist. | price> |
R-C-2568 | Zotiraciclib CAS:1204918-72-8 | Zotiraciclib(TG02;SB1317)is a potent inhibitor of CDK2,JAK2,and FLT3 for the treatment of cancer,with IC50s of 13,73,and 56 nM for CDK2,JAK2 and FLT3,respectively. | price> |
R-C-2668 | AG-14361 CAS:328543-09-5 | AG14361 is a potent PARP-1 inhibitor,with a Ki of < 5nM,and in permeabilized SW620 and intact SW620 cells,the IC50s are 29nM and 14nM,respectively. | price> |
R-C-2688 | TCS HDAC6 20b CAS:956154-63-5 | TCS HDAC6 20b,selective inhibitor of histone deacetylase 6(HDAC6).Inhibits HCT116 growth in combination with taxol. Also inhibits growth of MCF-7 cells stimulated by estrogen. | price> |
R-R-4368 | Ro 10-5824 dihydrochloride CAS No.189744-94-3 | Ro 10-5824 dihydrochloride/CAS No.189744-94-3 is a selective dopamine D4 receptor partial agonist, with Ki of 5.2 nM. | price> |