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Catalog	name	Description	price
R-C-2357	Protionamide CAS:14222-60-7	Protionamide(or prothionamide)is a drug used in the treatment of tuberculosis; has also been tested for use in the treatment of leprosy.Target:Anti tuberculosisAlthough ETH and PTH are both potent drugs against M.tuberculosis (MIC=～0.5μg/ml)(24),they do not affect E.coli growth,even at very high concentrations(100μg/ml),which is primarily caused by the absence of an EthA homologue in E.coli.	price>
R-R-4057	Apelin-36(rat, mouse) CAS No.230299-95-3	Apelin-36(rat, mouse)/CAS No.230299-95-3 is an endogenous orphan G protein-coupled receptor APJ agonist. Apelin-36(rat, mouse) binds to APJ receptors with an IC50 of 5.4 nM, and potently inhibits cAMP production with an EC50 of 0.52 nM. Apelin-36(rat, mouse) blocks entry of some HIV-1 and HIV-2 strains into NP-2/CD4 cells expressing APJ.	price>
R-C-2358	Taxifolin 7-O-rhamnoside	Taxifolin 7-O-rhamnoside(Taxifolin 7-O-α-L-rhamnoside)is a flavonoid isolated from Hypericum japonicum.	price>
R-R-4058	Bombesin CAS No.31362-50-2	Bombesin/CAS No.31362-50-2, a tetradecapeptide, plays an important role in the release of gastrin and the activation of G-protein receptors.	price>
R-C-2359	Steviolbioside CAS:41093-60-1	Steviolbioside is a rare sweetener that exists in stevia rebaudiana leaves. Steviolbioside presents inhibition on several human cancer cells and acts as potential remedy for human breast cancer.	price>
R-R-4059	PD176252 CAS No.204067-01-6	PD176252/CAS No.204067-01-6 is a potent antagonist of neuromedin-B preferring (BB1) and gastrin-releasing peptide-preferring (BB2) receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 nM for Rat BB1 and BB2 receptors, respectively; PD176252 is also an agonist of N-Formyl peptide receptor1/2 (FPR1/FPR2), with EC50s of 0.31 and 0.66 μM in HL-60 cells.	price>
R-C-2360	KKL-10 CAS:952849-76-2	KKL-10 is a small-molecule ribosome rescue inhibitor with broad-spectrum antimicrobial activity against bacteria.	price>
R-R-4060	MK-5046 CAS No.1022152-70-0	MK-5046/CAS No.1022152-70-0 is a potent, selective and orally active Bombesin receptor subtype-3 (BRS-3) allosteric agonist with an IC50 and an EC50 value of 27 and 25 nM for hBRS-3, respectively. MK-5046 inhibits food intake and reduces body weight of diet-induced obese (DIO) mouse models. MK-5046 can be used for the research of obesity.	price>
R-C-2361	Auranofin CAS:34031-32-8	Auranofin (Ridaura,SKF-39162)is an inhibitor of thioredoxin reductase(TrxR)with IC50 of 88 nM for purified H.pylori TrxR in cell-free assay.Auranofin has anti-cancer activity and can completely inhibit bacterial growth at 1.2μM.	price>
R-R-4061	RC-3095 TFA CAS No.1217463-61-0	RC-3095 TFA/CAS No.1217463-61-0 is a selective bombesin/gastrin releasing peptide receptor (GRPR) antagonist. RC-3095 TFA exerts protective effects by reducing gastric oxidative injury in the arthritic mice.	price>
R-C-2362	Aminothiazole CAS:96-50-4	Aminothiazole(2-Aminothiazole),a typical heterocyclic amine,is a precursor for the synthesis of biologically active molecules including sulfur agents,biocides, fungicides,antibiotics,dyes and chemical reaction accelerators.	price>
R-R-4062	ML-18 CAS No.1422269-30-4	ML-18/CAS No.1422269-30-4 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.	price>
R-C-2363	Fosfomycin calcium CAS:26472-47-9	Fosfomycin(phosphomycin,phosphonomycin)is bactericidal and inhibits bacterial cell wall biogenesis by inactivating the enzyme UDP-N-acetylglucosamine-3-enolpyruvyltransferase,also known as MurA.It enters the bacterial cell through the glycerophosphate transporter.	price>
R-R-4063	BIM 23042 TFA	BIM 23042 TFA, a certain somatostatin (SS) octapeptide analogue, is a selective neuropeptide neuromedin B receptor (NMB-R, BB1) antagonist. BIM 23042 has 100-fold lower affinity for gastrin-releasing peptide (GRP) receptor (BB2). BIM 23042 inhibits Neuromedin B (HY-P0241), ICI 216140 and DPDM-bombesin ethylamide-induced Ca2+ release.	price>
R-C-2364	Closantel CAS:57808-65-8	Closantel is a halogenated salicylanilide with a potent anti-parasitic activity.Closantel is a potent and highly specific Onchocerca volvulus chitinase(OvCHT1)inhibitor with an IC50 of 1.6μM and a Ki of 468nM.Closantel inhibits the O.volvulus L3 to L4 molt of developing.	price>
R-R-4064	PD 168368 CAS No.204066-82-0	PD 168368/CAS No.204066-82-0 is a potent, competitive, and selective neuromedin B receptor (NMB-R) antagonist with the Ki of 15–45 nM. PD 168368 is neuromedin B receptor (NMBR; IC50=96 nM) / gastrin-releasing peptide receptor (GRPR IC50=3500 nM) antagonist. PD 168368 also is a mixed FPR1/FPR2/FPR3 agonist with EC50s of 0.57, 0.24, and 2.7 nM, respectively.	price>
R-C-2365	Ftaxilide CAS:19368-18-4	Ftaxilide is a bioactive chemical.	price>
R-R-4065	Kuwanon G CAS No.75629-19-5	Kuwanon G/CAS No.75629-19-5 is a flavonoid isolated from Morus alba, acts as a bombesin receptor antagonist, with potential antimicrobial activity.	price>
R-C-2366	Pasiniazid CAS:2066-89-9	Pasiniazid is a biochemical used in the treatment of tuberculosis.	price>
R-R-4066	Kuwanon H CAS No.76472-87-2	Kuwanon H/CAS No.76472-87-2 is a flavonoid isolated from Morus alba, which acts as a potent non-peptide bombesin receptor antagonist. Kuwanon H selectively inhibits binding of gastrin releasing peptide CRP to GRP-preferring recepotr, with a Ki value of 290 nM in cells.	price>

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